SCHEMBL6493365

SCHEMBL6493365

Cc1c(F)ccc2c([C@@H]3CCN[C@@H](C)C3)c[nH]c12

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 13/20 0.44
APP P05067 3/20 0.37
AR P10275 1/20 0.36
HTR1A P08908 1/20 0.33
DRD1 P21728 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTR1B P28222 1/20 0.33
HTR2A P28223 1/20 0.33
SLC6A3 Q01959 1/20 0.33
PLG P00747 1/20 0.33
HTR2C P28335 2/20 0.32
ADRB2 P07550 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6491454 1.00 SLC6A4 (0.44) SLC6A4APPARHTR1ADRD1
SCHEMBL6502093 0.88 SLC6A4 (0.45) SLC6A4APPARHTR1ADRD1
SCHEMBL6501499 0.88 SLC6A4 (0.45) SLC6A4APPARHTR1ADRD1
SCHEMBL6491329 0.75 SLC6A4 (0.63) SLC6A4APPHTR1ADRD1SLC6A2
SCHEMBL6489351 0.75 SLC6A4 (0.63) SLC6A4APPHTR1ADRD1SLC6A2
SCHEMBL6492379 0.74 SLC6A4 (0.38) SLC6A4APPARHTR1AHTR1B
SCHEMBL8631277 0.71 HTR2C (0.65) SLC6A4HTR2AHTR2CADRB2
SCHEMBL6812125 0.69 APP (0.53) SLC6A4APPARHTR1ASLC6A2
SCHEMBL6499536 0.68 AR (0.44) ARHTR2A
SCHEMBL8819067 0.65 SLC6A4 (0.46) SLC6A4HTR1ADRD1SLC6A2HTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6844338-B2 Piperidyindoles as serotonin receptor ligands ELI LILLY AND COMPANY (US) 2005-01-18 US disclosed
US-20030225068-A1 Piperidyindoles as serotonin receptor ligands ELI LILLY AND COMPANY 2003-12-04 US disclosed
EP-1286992-A1 PIPERIDYINDOLES AS SEROTONIN RECEPTOR LIGANDS ELI LILLY AND COMPANY (US) 2003-03-05 EP disclosed
WO-2001087881-A1 PIPERIDYINDOLES AS SEROTONIN RECEPTOR LIGANDS ELI LILLY AND COMPANY (US) 2001-11-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225068-A1 Piperidyindoles as serotonin receptor ligands CNR1, HTR1D, HTR1A SLC6A4 215/4885APP 2484/4885AR 299/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.