SCHEMBL6497667

SCHEMBL6497667

CC(NC(=O)C1CCN(C(=O)C=Cc2cc(C(F)(F)F)ccc2F)CC1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.48
ENPP2 Q13822 7/20 0.46
CAPN1 P07384 3/20 0.42
BACE1 P56817 1/20 0.41
KCNH2 Q12809 2/20 0.41
KMT2A Q03164 2/20 0.41
TEAD1 P28347 2/20 0.40
C3AR1 Q16581 1/20 0.40
MEN1 O00255 1/20 0.40
TSHR P16473 1/20 0.40
ITGAL P20701 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6497665 1.00 SMN1; SMN2 (0.48) SMN1; SMN2ENPP2CAPN1BACE1KCNH2
SCHEMBL6504860 0.91 ENPP2 (0.46) SMN1; SMN2ENPP2CAPN1KCNH2KMT2A
SCHEMBL6495356 0.90 ENPP2 (0.46) ENPP2CAPN1KCNH2KMT2ATEAD1
SCHEMBL6495354 0.90 ENPP2 (0.46) ENPP2CAPN1KCNH2KMT2ATEAD1
SCHEMBL6500473 0.87 SMN1; SMN2 (0.66) SMN1; SMN2CAPN1KMT2AC3AR1MEN1
SCHEMBL6500476 0.87 SMN1; SMN2 (0.66) SMN1; SMN2CAPN1KMT2AC3AR1MEN1
SCHEMBL6497183 0.84 ITGAL (0.45) SMN1; SMN2ENPP2CAPN1KMT2AMEN1
SCHEMBL6497179 0.84 ITGAL (0.45) SMN1; SMN2ENPP2CAPN1KMT2AMEN1
SCHEMBL6504618 0.83 CAPN1 (0.46) SMN1; SMN2CAPN1KMT2AC3AR1MEN1
SCHEMBL6504616 0.83 CAPN1 (0.46) SMN1; SMN2CAPN1KMT2AC3AR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO claimed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed