SCHEMBL6497889

SCHEMBL6497889

[CH2]C(=O)NC1CCCNC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.47
OPRK1 P41145 1/20 0.47
SLC6A1 P30531 2/20 0.44
SLC6A11 P48066 1/20 0.44
TSHR P16473 1/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
SLC6A13 Q9NSD5 1/20 0.44
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
CYP2D6 P10635 1/20 0.42
PBK Q96KB5 4/20 0.42
EPHX1 P07099 1/20 0.41
CHRNA1 P02708 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA4 P43681 1/20 0.40
CHEK1 O14757 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3314984 0.88
SCHEMBL148965 0.82 SLC6A1 (0.50) MAPK1OPRK1SLC6A1SLC6A11TSHR
SCHEMBL1968950 0.82 SLC6A1 (0.50) MAPK1OPRK1SLC6A1SLC6A11TSHR
SCHEMBL475548 0.82 SLC6A1 (0.50) MAPK1OPRK1SLC6A1SLC6A11TSHR
SCHEMBL23139818 0.80 MAPK1 (0.47) MAPK1OPRK1SLC6A1SLC6A11TSHR
SCHEMBL1006531 0.80 MAPK1 (0.50) MAPK1OPRK1SLC6A1SLC6A11TSHR
SCHEMBL17902608 0.80 MAPK1 (0.47) MAPK1OPRK1SLC6A1SLC6A11TSHR
SCHEMBL16561741 0.80 KDM4E (0.52) MAPK1OPRK1SLC6A1SLC6A11KDM4E
SCHEMBL12260711 0.80 EPHX1 (0.66) MAPK1OPRK1SLC6A1SLC6A11TSHR
Hydrochloric Acid SCHEMBL17560394 0.80 SLC6A1 (0.48) MAPK1OPRK1SLC6A1SLC6A11TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO claimed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed