SCHEMBL650135

SCHEMBL650135

COc1ccc(N=C2NC(=O)C(=Cc3cnc(NC(=O)C4CC4)s3)S2)c(C(=O)O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.43
GSK3B P49841 1/20 0.41
AKR1B1 P15121 1/20 0.40
DAPK3 O43293 1/20 0.40
DYRK3 O43781 1/20 0.40
PIM1 P11309 1/20 0.40
CSNK2A1 P68400 1/20 0.40
DYRK1A Q13627 1/20 0.40
PIM3 Q86V86 1/20 0.40
HIPK2 Q9H2X6 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
CSNK1G1 Q9HCP0 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
MAPT P10636 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
PTPN11 Q06124 1/20 0.39
ALOX15 P16050 1/20 0.39
PTGS2 P35354 1/20 0.39
HSD11B1 P28845 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL651308 1.00 ABL1 (0.43) ABL1GSK3BAKR1B1DAPK3DYRK3
SCHEMBL10176547 0.90 MAPT (0.47) ABL1GSK3BAKR1B1DAPK3DYRK3
SCHEMBL697898 0.85 MAPT (0.43) ABL1GSK3BAKR1B1DYRK1AMAPT
SCHEMBL651724 0.85 PTPN7 (0.44) MAPTMEN1KMT2APTPN11HSD11B1
SCHEMBL10176532 0.83 PTPN7 (0.44) ABL1MAPTMEN1KMT2APTPN11
SCHEMBL652132 0.82 MAPT (0.55) ABL1MAPTMEN1KMT2AALOX15
SCHEMBL653891 0.82 MAPT (0.41) ABL1MAPTMEN1KMT2ALMNA
SCHEMBL653892 0.82 MAPT (0.41) ABL1MAPTMEN1KMT2ALMNA
SCHEMBL703259 0.81 MEN1 (0.38) MAPTMEN1KMT2APTPN11HSD11B1
SCHEMBL650134 0.81 AKR1B1 (0.39) AKR1B1DAPK3DYRK3PIM1CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423204-A1 THIAZOLIDINONE DERIVATIVE SBI Biotech Co., Ltd. (JP) 2012-02-29 EP disclosed
US-8119812-B2 Thiazolidinone derivative SBI BIOTECH CO., LTD. (JP) 2012-02-21 US disclosed
US-20110190299-A1 THIAZOLIDINONE DERIVATIVE SBI BIOTECH CO., LTD. (JP) 2011-08-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110190299-A1 THIAZOLIDINONE DERIVATIVE CDC7, CDK17, CDCA2 ABL1 978/4885GSK3B 305/4885AKR1B1 1750/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.