SCHEMBL6501467

SCHEMBL6501467

CC(C)CC(=O)Nc1nc(-c2ccccc2)cc(-c2ccccc2)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 14/20 1.00
ADORA3 P0DMS8 8/20 0.71
ADORA2A P29274 4/20 0.71
ADORA2B P29275 1/20 0.71
SMN1; SMN2 Q16637 3/20 0.53
KDM4E B2RXH2 1/20 0.53
MAPT P10636 1/20 0.53
HTT P42858 1/20 0.53
GAA P10253 1/20 0.51
RAB9A P51151 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26053899 0.84 ADORA1 (0.72) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL6505603 0.83 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BKDM4E
SCHEMBL26053924 0.83 ADORA1 (0.71) ADORA1ADORA3ADORA2AADORA2BSMN1; SMN2
SCHEMBL16391805 0.82 ADORA1 (0.72) ADORA1ADORA3ADORA2AADORA2BSMN1; SMN2
SCHEMBL4829224 0.82 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BSMN1; SMN2
SCHEMBL6499771 0.81 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BKDM4E
SCHEMBL24227646 0.80 ADORA1 (0.72) ADORA1ADORA3ADORA2AADORA2BMAPT
SCHEMBL6502989 0.80 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL24227492 0.79 ADORA1 (0.76) ADORA1ADORA3ADORA2AADORA2BKDM4E
SCHEMBL26055757 0.78 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033085-A1 PYRIMIDINES DERIVATIVES AS ADENOSINE RECEPTORS LIGANDS UNIVERSITEIT LEIDEN (NL) 2005-04-14 WO claimed
WO-2005033085-A1 PYRIMIDINES DERIVATIVES AS ADENOSINE RECEPTORS LIGANDS UNIVERSITEIT LEIDEN (NL) 2005-04-14 WO disclosed