SCHEMBL6502989

SCHEMBL6502989

CC(C)C(=O)Nc1nc(-c2ccccc2)cc(-c2ccccc2)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 17/20 1.00
ADORA3 P0DMS8 6/20 0.69
ADORA2A P29274 5/20 0.67
ADORA2B P29275 1/20 0.63
NOS1 P29475 1/20 0.56
TDP1 Q9NUW8 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19699609 0.84 ADORA1 (0.73) ADORA1ADORA3ADORA2ANOS1
SCHEMBL6497567 0.83 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL26053899 0.82 ADORA1 (0.72) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL26055757 0.81 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BTDP1
SCHEMBL6529699 0.81 ADORA1 (0.74) ADORA1ADORA3ADORA2AADORA2BTDP1
SCHEMBL16391790 0.81 ADORA1 (0.70) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL4822464 0.80 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL6501467 0.80 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL26053924 0.78 ADORA1 (0.71) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL6507291 0.77 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033085-A1 PYRIMIDINES DERIVATIVES AS ADENOSINE RECEPTORS LIGANDS UNIVERSITEIT LEIDEN (NL) 2005-04-14 WO claimed
US-20230271983-A1 FUNCTIONALIZED ISONITRILES AND PRODUCTS, PREPARATION AND USES THEREOF UNIVERSIDADE DE SANTIAGO DE COMPOSTELA (ES) 2023-08-31 US disclosed
US-20230271983-A1 FUNCTIONALIZED ISONITRILES AND PRODUCTS, PREPARATION AND USES THEREOF UNIVERSIDADE DE SANTIAGO DE COMPOSTELA (ES) 2023-08-31 US disclosed
US-20050272740-A1 Benzimidazole derivatives MERCK PATENT GMBH (DE) 2005-12-08 US disclosed
WO-2005033085-A1 PYRIMIDINES DERIVATIVES AS ADENOSINE RECEPTORS LIGANDS UNIVERSITEIT LEIDEN (NL) 2005-04-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050272740-A1 Benzimidazole derivatives F12, F11, SERPINC1 ADORA1 572/4885ADORA3 778/4885ADORA2A 2033/4885
US-20230271983-A1 FUNCTIONALIZED ISONITRILES AND PRODUCTS, PREPARATION AND USES THEREOF KIT, MACF1, IK ADORA1 1360/4885ADORA3 1458/4885ADORA2A 2807/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.