SCHEMBL6501679

SCHEMBL6501679

Cc1ccc(S(=O)(=O)NC(=O)c2cc(C)c3nc(C)n(Cc4ccc(N(C)C(=O)OC(C)(C)C)cc4Cl)c3n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT8 Q9H7Z6 2/20 0.39
KAT6A Q92794 2/20 0.39
KAT5 Q92993 2/20 0.39
PTGS2 P35354 2/20 0.35
PTGS1 P23219 1/20 0.35
F2 P00734 1/20 0.34
FLT1 P17948 3/20 0.33
FLT4 P35916 3/20 0.33
KDR P35968 3/20 0.33
KDM4E B2RXH2 1/20 0.33
EGFR P00533 1/20 0.33
ALKBH2 Q6NS38 1/20 0.32
ALKBH5 Q6P6C2 1/20 0.32
ALKBH3 Q96Q83 1/20 0.32
FTO Q9C0B1 1/20 0.32
HSD17B13 Q7Z5P4 1/20 0.32
PPARG P37231 2/20 0.32
RAB9A P51151 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
NR2E3 Q9Y5X4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6491998 0.91 F2 (0.36) KAT8KAT6AKAT5PTGS2PTGS1
SCHEMBL6502253 0.89 KAT8 (0.39) KAT8KAT6AKAT5PTGS2PTGS1
SCHEMBL6504184 0.86 PTGS2 (0.38) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL6497677 0.86 PPARG (0.47) PPARG
SCHEMBL6494878 0.85 PTGS2 (0.37) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL6499896 0.85 NQO2 (0.35) KAT8KAT6AKAT5HSD17B13RAB9A
SCHEMBL6500370 0.84 PIK3CB (0.37) KAT8KAT6AKAT5HSD17B13PPARG
SCHEMBL6298633 0.82 FLT1 (0.42) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL6299098 0.82 PPARG (0.44) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL6299197 0.81 FLT1 (0.41) PTGS2PTGS1FLT1FLT4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030171396-A1 Sulfonamide compounds and uses thereof as medicines FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2003-09-11 US claimed
US-6573274-B1 Treatment of the diseases curable based on a hypoglycemic action, and the diseases curable based on a cGMP-PDE inhibitory action, a smooth muscle relaxing action, a bronchodilating action, a vasodilating action, a smooth muscle FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2003-06-03 US claimed
EP-1136492-A1 SULFONAMIDE COMPOUNDS AND USES THEREOF AS MEDICINES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-09-26 EP claimed
US-6890934-B2 Sulfonamide compounds and uses thereof as medicines FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-05-10 US disclosed
US-20030171396-A1 Sulfonamide compounds and uses thereof as medicines FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2003-09-11 US disclosed
US-6573274-B1 Treatment of the diseases curable based on a hypoglycemic action, and the diseases curable based on a cGMP-PDE inhibitory action, a smooth muscle relaxing action, a bronchodilating action, a vasodilating action, a smooth muscle FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2003-06-03 US disclosed
EP-1136492-A1 SULFONAMIDE COMPOUNDS AND USES THEREOF AS MEDICINES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-09-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030171396-A1 Sulfonamide compounds and uses thereof as medicines PDE2A, PDE3A, PDE5A KAT8 4148/4885KAT6A 4278/4885KAT5 3636/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.