SCHEMBL6502673

SCHEMBL6502673

CSc1cccc(-c2cc(CN(CCO)CCO)c(=O)n(CC(C)C)n2)c1

nearest known ligand 0.32

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DYRK3 O43781 1/20 0.32
CCNT1 O60563 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CDK9 P50750 1/20 0.32
CDK5 Q00535 1/20 0.32
DYRK1A Q13627 1/20 0.32
CDK5R1 Q15078 1/20 0.32
DYRK2 Q92630 1/20 0.32
DYRK1B Q9Y463 1/20 0.32
KDM4E B2RXH2 1/20 0.31
BACE1 P56817 2/20 0.31
IDO1 P14902 1/20 0.31
TGFBR1 P36897 1/20 0.31
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30
KEAP1 Q14145 1/20 0.30
NFE2L2 Q16236 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL6491090 0.96 AKR1C3 (0.32) DYRK3CCNT1CCNA2CDK2CDK9
SCHEMBL1925562 0.89 ADORA3 (0.34)
SCHEMBL1925331 0.87 KDM4E (0.38) KDM4E
Hydrochloric Acid SCHEMBL1927907 0.86 KDM4E (0.37) KDM4E
Oxalic Acid SCHEMBL1924390 0.85 ADORA3 (0.34)
SCHEMBL1924826 0.85 MEN1 (0.38) KDM4E
Hydrochloric Acid SCHEMBL1927605 0.84 MEN1 (0.37) KDM4E
Hydrochloric Acid SCHEMBL6502437 0.83 MEN1 (0.39) KDM4E
SCHEMBL1924523 0.82 HTT (0.34)
SCHEMBL1924759 0.81 MEN1 (0.40) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6861428-B2 Water-soluble phenylpyridazine compounds and compositions containing the same KOWA CO., LTD. (JP) 2005-03-01 US disclosed