SCHEMBL6503495

SCHEMBL6503495

COC(=O)C(CCSC)NC(=O)C1CCN(C(=O)/C=C/c2ccc(SC)c(Cl)c2Cl)CC1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGAL P20701 7/20 0.49
ITGB2 P05107 6/20 0.49
ICAM1 P05362 6/20 0.49
CAPN1 P07384 4/20 0.43
TSHR P16473 1/20 0.41
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ENPP2 Q13822 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6503498 1.00 ITGAL (0.49) ITGALITGB2ICAM1CAPN1TSHR
SCHEMBL8297244 1.00 ITGAL (0.49) ITGALITGB2ICAM1CAPN1TSHR
SCHEMBL8298603 0.92 ITGAL (0.49) ITGALITGB2ICAM1CAPN1KDM4E
SCHEMBL6506580 0.92 ITGAL (0.49) ITGALITGB2ICAM1CAPN1KDM4E
SCHEMBL6506577 0.92 ITGAL (0.49) ITGALITGB2ICAM1CAPN1KDM4E
SCHEMBL6497005 0.92 ITGB2 (0.50) ITGALITGB2ICAM1CAPN1TSHR
SCHEMBL8297179 0.92 ITGB2 (0.50) ITGALITGB2ICAM1CAPN1TSHR
SCHEMBL6497008 0.92 ITGB2 (0.50) ITGALITGB2ICAM1CAPN1TSHR
SCHEMBL8296890 0.90 ITGAL (0.50) ITGALITGB2ICAM1CAPN1KDM4E
SCHEMBL8298637 0.89 CAPN1 (0.53) ITGALITGB2ICAM1CAPN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed