SCHEMBL8298637

SCHEMBL8298637

COC(=O)[C@H](CC(C)C)NC(=O)C1CCN(C(=O)/C=C/c2ccc(SC)c(Cl)c2Cl)CC1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 4/20 0.53
ITGAL P20701 8/20 0.49
ITGB2 P05107 7/20 0.49
ICAM1 P05362 7/20 0.49
NOS3 P29474 3/20 0.45
NOS1 P29475 3/20 0.45
NOS2 P35228 3/20 0.45
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ENPP2 Q13822 1/20 0.38
MAPK1 P28482 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6499090 0.91 CAPN1 (0.54) CAPN1ITGALITGB2ICAM1MAPK1
SCHEMBL6499094 0.91 CAPN1 (0.54) CAPN1ITGALITGB2ICAM1MAPK1
SCHEMBL8296890 0.91 ITGAL (0.50) CAPN1ITGALITGB2ICAM1KDM4E
SCHEMBL8298603 0.89 ITGAL (0.49) CAPN1ITGALITGB2ICAM1KDM4E
SCHEMBL6506580 0.89 ITGAL (0.49) CAPN1ITGALITGB2ICAM1KDM4E
SCHEMBL6506577 0.89 ITGAL (0.49) CAPN1ITGALITGB2ICAM1KDM4E
SCHEMBL6503498 0.89 ITGAL (0.49) CAPN1ITGALITGB2ICAM1KDM4E
SCHEMBL6503495 0.89 ITGAL (0.49) CAPN1ITGALITGB2ICAM1KDM4E
SCHEMBL8297244 0.89 ITGAL (0.49) CAPN1ITGALITGB2ICAM1KDM4E
SCHEMBL6533299 0.89 ITGAL (0.53) CAPN1ITGALITGB2ICAM1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed