SCHEMBL6506341

SCHEMBL6506341

COC(=O)C(Cc1cnc2ccccc2c1)NC(=O)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.45
MDM4 O15151 2/20 0.44
TP53 P04637 2/20 0.44
TGM2 P21980 2/20 0.43
ITGA4 P13612 1/20 0.43
ITGB7 P26010 1/20 0.43
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
MMP8 P22894 1/20 0.42
CASP3 P42574 1/20 0.41
MDM2 Q00987 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6506337 1.00 SIRT2 (0.45) SIRT2MDM4TP53TGM2ITGA4
SCHEMBL29679135 0.91 MDM4 (0.51) MDM4TP53TGM2ITGA4ITGB7
SCHEMBL6499392 0.91 MDM4 (0.51) MDM4TP53TGM2ITGA4ITGB7
SCHEMBL119871 0.91 MDM4 (0.51) MDM4TP53TGM2ITGA4ITGB7
SCHEMBL6499381 0.91 MDM4 (0.51) MDM4TP53TGM2ITGA4ITGB7
SCHEMBL15697341 0.85 CTSB (0.49) MDM4TP53CASP3
SCHEMBL17054211 0.82 MDM4 (0.45) MDM4TP53CASP3MDM2
SCHEMBL2977877 0.82 ATM (0.53) MDM4TP53CASP3
SCHEMBL12531899 0.82 ATM (0.53) MDM4TP53CASP3
SCHEMBL13743302 0.82 ATM (0.53) MDM4TP53CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed