SCHEMBL6506438

SCHEMBL6506438

CN1C(=O)Cc2cc(Cn3ccc(OCc4ccc(F)cc4F)c(Cl)c3=O)ccc21

nearest known ligand 0.52

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 19/20 0.52
PTGER1 P34995 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6474630 0.85 MAPK14 (0.62) MAPK14
SCHEMBL4473803 0.82 MAPK14 (0.55) MAPK14
SCHEMBL4476599 0.81 MAPK14 (0.52) MAPK14
SCHEMBL4471766 0.81 MAPK14 (0.49) MAPK14
SCHEMBL4468144 0.81 MAPK14 (0.49) MAPK14
SCHEMBL6471669 0.81 MAPK14 (0.52) MAPK14
SCHEMBL4375353 0.81 MAPK14 (0.60) MAPK14
SCHEMBL4474437 0.81 MAPK14 (0.52) MAPK14PTGER1
SCHEMBL4468176 0.81 MAPK14 (0.52) MAPK14
SCHEMBL6533880 0.80 MAPK14 (0.43) MAPK14PTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050176775-A1 Substituted pyridinones PHARMACIA CORPORATION 2005-08-11 US claimed
US-20050176775-A1 Substituted pyridinones PHARMACIA CORPORATION 2005-08-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050176775-A1 Substituted pyridinones MAPK1, MAPK6, MAP3K6 MAPK14 53/4885PTGER1 102/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.