SCHEMBL6507067

SCHEMBL6507067

[NH]C(=O)c1nc(-c2ccc(C(F)(F)F)cc2)oc1-c1ccc2ccccc2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.46
AR P10275 2/20 0.40
HSPD1 P10809 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPN5 P54829 1/20 0.39
HSPE1 P61604 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2D6 P10635 1/20 0.38
PDE10A Q9Y233 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6507069 0.89 IKBKB (0.58) IKBKBARHSPD1PTPN2PTPN1
SCHEMBL6510847 0.81 NPC1 (0.43) IKBKBHDAC3HDAC1HDAC2HDAC8
SCHEMBL6365995 0.77 FTO (0.46) PTPN1PPARG
SCHEMBL6365992 0.77 FTO (0.46) PTPN1PPARG
SCHEMBL6366531 0.76 MCL1 (0.40) IKBKBPTPN1CYP3A4PPARGP2RY14
SCHEMBL6366525 0.76 MCL1 (0.40) IKBKBPTPN1CYP3A4PPARGP2RY14
SCHEMBL6365927 0.75 CDK2 (0.45) PTPN1P2RY14
SCHEMBL6365922 0.75 CDK2 (0.45) PTPN1P2RY14
SCHEMBL22734790 0.73 NPC1 (0.62) ARNPC1RAB9ACYP1A2CYP2C19
SCHEMBL29544777 0.73 NPC1 (0.62) ARNPC1RAB9ACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005113522-A1 AZOLE CARBOXAMIDE INHIBITORS OF BACTERIAL TYPE III PROTEIN SECRETION SYSTEMS JANSSEN PHARMACEUTICA, N.V. (BE) 2005-12-01 WO disclosed