SCHEMBL6507215

SCHEMBL6507215

NC(=O)Nc1sc(NC(=O)c2cccc(CN3CCCCC3)c2)cc1C(N)=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.62
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
HIF1A Q16665 1/20 0.50
KDM4E B2RXH2 3/20 0.47
MAPT P10636 3/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
HPGD P15428 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
RAB9A P51151 4/20 0.47
HTT P42858 2/20 0.47
GAA P10253 1/20 0.47
NPC1 O15118 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
PARP1 P09874 2/20 0.42
GLS O94925 1/20 0.42
IKBKB O14920 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6510633 0.82 MEN1 (0.48) CHEK1KDM4EMAPTMEN1KMT2A
SCHEMBL6512362 0.77 IKBKB (0.57) MAPTMEN1KMT2ARAB9AGAA
SCHEMBL1926828 0.77 CHEK1 (1.00) CHEK1KDM4EMAPTMEN1KMT2A
SCHEMBL6506340 0.76 FLT3 (0.51) KDM4EMAPTMEN1KMT2AHPGD
SCHEMBL1928372 0.76 CHEK1 (0.98) CHEK1KDM4EMAPTMEN1KMT2A
SCHEMBL6530168 0.75 IKBKB (0.62) CHEK1MAPTMEN1KMT2ANPSR1
SCHEMBL1397213 0.75 CYP2D6 (0.75) CYP2D6CYP2C9HIF1AKDM4EGAA
SCHEMBL6507704 0.74 CHEK1 (0.49) CHEK1KDM4EMAPTMEN1KMT2A
SCHEMBL6510003 0.74 P2RX1 (0.52) MAPTMEN1KMT2ARAB9AHTT
SCHEMBL6583311 0.74 CYP2D6 (0.68) CYP2D6CYP2C9HIF1AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed