SCHEMBL6507291

SCHEMBL6507291

CC(C)(C)C(=O)Nc1nc(-c2ccccc2)cc(-c2ccccc2)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 15/20 1.00
ADORA3 P0DMS8 5/20 0.69
ADORA2A P29274 3/20 0.63
ADORA2B P29275 1/20 0.63
POLB P06746 1/20 0.60
TDP1 Q9NUW8 1/20 0.54
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26055757 0.81 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BTDP1
SCHEMBL6529699 0.81 ADORA1 (0.74) ADORA1ADORA3ADORA2AADORA2BTDP1
SCHEMBL4824825 0.80 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BPOLB
SCHEMBL6505603 0.77 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BMEN1
SCHEMBL6502989 0.77 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2BTDP1
SCHEMBL6498848 0.77 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL13040786 0.77 ADORA1 (0.61) ADORA1ADORA3ADORA2AADORA2BPOLB
SCHEMBL3451038 0.76 ADORA1 (0.61) ADORA1ADORA3ADORA2AADORA2BTDP1
SCHEMBL13040784 0.76 ADORA1 (0.60) ADORA1ADORA3ADORA2AADORA2BPOLB
SCHEMBL6499771 0.75 ADORA1 (1.00) ADORA1ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033085-A1 PYRIMIDINES DERIVATIVES AS ADENOSINE RECEPTORS LIGANDS UNIVERSITEIT LEIDEN (NL) 2005-04-14 WO claimed
WO-2005033085-A1 PYRIMIDINES DERIVATIVES AS ADENOSINE RECEPTORS LIGANDS UNIVERSITEIT LEIDEN (NL) 2005-04-14 WO disclosed
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO disclosed