SCHEMBL6507679

SCHEMBL6507679

Nc1cccc(-c2ccnc(NC(=O)O)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.54
CNR1 P21554 1/20 0.49
WNT3A P56704 1/20 0.48
MAP4K4 O95819 1/20 0.47
MAOA P21397 1/20 0.46
PIK3C3 Q8NEB9 8/20 0.45
KARS1 Q15046 1/20 0.45
MCL1 Q07820 1/20 0.44
GSK3B P49841 1/20 0.44
PIP5K1C O60331 1/20 0.44
PIK3CA P42336 1/20 0.44
FDPS P14324 1/20 0.43
MAPK8 P45983 1/20 0.43
MAPK10 P53779 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17872892 0.85 EGFR (0.69) EGFRCNR1WNT3APIK3C3GSK3B
SCHEMBL17631827 0.83 MKNK1 (0.53) EGFRCNR1WNT3APIK3C3MAPK8
SCHEMBL17010231 0.82 NR3C2 (0.44) EGFRPIK3C3
SCHEMBL6507708 0.81 PIP5K1C (0.63) EGFRCNR1WNT3APIP5K1CPIK3CA
SCHEMBL6502882 0.80 IRAK4 (0.49) EGFRMAP4K4PIK3C3GSK3B
SCHEMBL1026072 0.79 FFAR1 (0.47) PIK3CA
SCHEMBL1026728 0.78 NR3C2 (0.64) MAOA
SCHEMBL6508127 0.77 CGAS (0.44) EGFRPIK3C3GSK3BMAPK8MAPK10
SCHEMBL6508122 0.77 CGAS (0.44) EGFRPIK3C3GSK3BMAPK8MAPK10
SCHEMBL17872874 0.74 KDM4E (0.51) EGFRCNR1WNT3AGSK3BMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003123-A1 NOVEL PYRIDINE DERIVATIVES AS JNK SPECIFIC INHIBITORS ASTRAZENECA AB (SE) 2005-01-13 WO disclosed