SCHEMBL6507970

SCHEMBL6507970

CCN(CCOc1ccccc1)Cc1ccc(-c2ccc(C(=O)O)s2)nc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 9/20 0.52
MAOB P27338 1/20 0.44
CYP1A2 P05177 1/20 0.44
LTA4H P09960 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44
CYP3A4 P08684 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ACKR3 P25106 3/20 0.42
NR4A2 P43354 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
IDH1 O75874 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6515011 0.93 HDAC1 (0.52) HDAC1MAOBCYP1A2LTA4HCYP2D6
SCHEMBL6509962 0.91 HDAC1 (0.65) HDAC1CYP3A4ACKR3
SCHEMBL6509511 0.86 HDAC1 (0.47) HDAC1CYP3A4KDM4ENR4A2ALDH1A1
SCHEMBL6513829 0.81 HDAC1 (0.65) HDAC1CYP3A4
SCHEMBL6531317 0.81 MAOB (0.43) MAOBCYP1A2LTA4HCYP2D6CYP2C9
SCHEMBL6509983 0.79 HDAC1 (0.76) HDAC1CYP3A4
SCHEMBL6514444 0.79 HPGD (0.42) HDAC1MAOBCYP1A2LTA4HCYP2D6
SCHEMBL6509316 0.78 HDAC1 (0.59) HDAC1HTTCYP3A4KDM4EACKR3
SCHEMBL8294397 0.78 HDAC1 (0.54) HDAC1CYP3A4ACKR3
SCHEMBL6512133 0.78 HDAC1 (0.61) HDAC1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005014588-A1 SUBSTITUTED THIENYL-HYDROXAMIC ACIDS HAVING HISTONE DEACETYLASE ACTIVITY ARGENTA DISCOVERY LIMITED (GB) 2005-02-17 WO disclosed