SCHEMBL6509316

SCHEMBL6509316

O=C(O)c1ccc(-c2ccc(CN(CCO)Cc3ccccc3)cn2)s1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 11/20 0.59
CYP3A4 P08684 1/20 0.51
KDM4E B2RXH2 1/20 0.48
ACKR3 P25106 5/20 0.45
HTT P42858 1/20 0.42
NR4A2 P43354 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6510513 0.90 HDAC1 (0.74) HDAC1CYP3A4ACKR3
SCHEMBL6510533 0.83 HDAC1 (0.67) HDAC1CYP3A4ACKR3
SCHEMBL6507970 0.78 HDAC1 (0.52) HDAC1CYP3A4KDM4EACKR3HTT
SCHEMBL6513829 0.78 HDAC1 (0.65) HDAC1CYP3A4
SCHEMBL6511673 0.76 HDAC1 (0.79) HDAC1CYP3A4ACKR3
SCHEMBL8294397 0.75 HDAC1 (0.54) HDAC1CYP3A4ACKR3
SCHEMBL8290112 0.74 HDAC1 (0.74) HDAC1CYP3A4ACKR3
SCHEMBL6509511 0.73 HDAC1 (0.47) HDAC1CYP3A4KDM4ENR4A2
SCHEMBL6515011 0.72 HDAC1 (0.52) HDAC1CYP3A4ACKR3HTT
SCHEMBL6507559 0.70 HDAC1 (0.69) HDAC1CYP3A4ACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005023762-A1 PYRROLIDINE-2-CARBONITRILE DERIVATIVES AND THEIR USE AS INHIBITORS OF DIPEPTIDYL PEPTIDASE-IV (DPP-IV) ABBOTT LABORATORIES (US) 2005-03-17 WO claimed
WO-2005014588-A1 SUBSTITUTED THIENYL-HYDROXAMIC ACIDS HAVING HISTONE DEACETYLASE ACTIVITY ARGENTA DISCOVERY LIMITED (GB) 2005-02-17 WO disclosed