SCHEMBL6509538

SCHEMBL6509538

CCN1CCN(c2cc(C)c3ccc(OC)cc3n2)CC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.70
ALDH1A1 P00352 9/20 0.70
HPGD P15428 4/20 0.70
CYP1A2 P05177 1/20 0.70
CYP2C19 P33261 1/20 0.70
MAPT P10636 11/20 0.67
NPSR1 Q6W5P4 1/20 0.67
L3MBTL1 Q9Y468 3/20 0.63
SMN1; SMN2 Q16637 2/20 0.63
TDP1 Q9NUW8 1/20 0.63
HSD17B10 Q99714 2/20 0.61
TSHR P16473 1/20 0.61
CASP1 P29466 1/20 0.61
AHR P35869 1/20 0.61
CASP7 P55210 1/20 0.61
TP53 P04637 1/20 0.57
RAD52 P43351 1/20 0.57
GAA P10253 2/20 0.56
NPC1 O15118 1/20 0.56
GLA P06280 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6512019 0.84 KDM4E (0.86) KDM4EALDH1A1HPGDCYP1A2CYP2C19
SCHEMBL6513981 0.81 KDM4E (0.70) KDM4EALDH1A1HPGDCYP1A2CYP2C19
SCHEMBL5910684 0.80 KMT2A (0.72) KDM4EALDH1A1HPGDMAPTL3MBTL1
SCHEMBL4215600 0.78 HRH3 (0.67) KDM4EALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL5909889 0.78 MAPT (0.86) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL5910416 0.75 POLB (0.82) KDM4EALDH1A1HPGDMAPTL3MBTL1
SCHEMBL6229712 0.75 ALDH1A1 (0.61) KDM4EALDH1A1HPGDCYP1A2CYP2C19
SCHEMBL5910106 0.74 MAPT (0.60) KDM4EALDH1A1HPGDMAPTL3MBTL1
SCHEMBL5909997 0.74 MCHR1 (0.84) KDM4EALDH1A1HPGDMAPTHSD17B10
Hydrochloric Acid SCHEMBL6231608 0.74 ALDH1A1 (0.60) KDM4EALDH1A1HPGDCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005087742-A1 METABOLIC KINASE MODULATORS AND METHODS OF USE AS PESTICIDES EXELIXIS, INC. (US) 2005-09-22 WO claimed
WO-2005087742-A1 METABOLIC KINASE MODULATORS AND METHODS OF USE AS PESTICIDES EXELIXIS, INC. (US) 2005-09-22 WO disclosed