SCHEMBL6509549

SCHEMBL6509549

O=C(O)CC(NC(=O)c1c(Cl)cncc1Cl)c1ccc(NC(=O)c2c(Cl)cncc2Cl)cc1

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 18/20 0.63
ITGA4 P13612 18/20 0.63
CTSA P10619 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6513196 0.91 ITGB1 (0.53) ITGB1ITGA4
SCHEMBL6509525 0.89 ITGB1 (0.52) ITGB1ITGA4CTSA
SCHEMBL6520277 0.89 ITGB1 (0.51) ITGB1ITGA4CTSA
SCHEMBL6518236 0.89 ITGB1 (0.52) ITGB1ITGA4CTSA
SCHEMBL6512380 0.88 ITGA4 (0.50) ITGB1ITGA4
SCHEMBL6518082 0.87 ITGB1 (0.57) ITGB1ITGA4
SCHEMBL6512395 0.87 ITGB1 (0.49) ITGB1ITGA4
SCHEMBL6514009 0.86 ITGB1 (0.58) ITGB1ITGA4
SCHEMBL6512464 0.86 SMN1; SMN2 (0.52) ITGB1ITGA4
SCHEMBL6513307 0.85 ITGB1 (0.48) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953798-B1 β-alanine derivates CELLTECH R&D LIMITED (GB) 2005-10-11 US claimed
EP-1135371-A1 BETA-ALANINE DERIVATIVES AS ALPHA 4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2001-09-26 EP claimed
WO-2000032575-A1 β-ALANINE DERIVATIVES AS α4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2000-06-08 WO claimed
US-6953798-B1 β-alanine derivates CELLTECH R&D LIMITED (GB) 2005-10-11 US disclosed
EP-1135371-A1 BETA-ALANINE DERIVATIVES AS ALPHA 4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2001-09-26 EP disclosed
WO-2000032575-A1 β-ALANINE DERIVATIVES AS α4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2000-06-08 WO disclosed