SCHEMBL6512177

SCHEMBL6512177

COC(=O)[C@H](Cc1ccc(NC(=O)c2c(F)cccc2F)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.53
ITGA4 P13612 4/20 0.53
ITGB3 P05106 1/20 0.52
ITGAV P06756 1/20 0.52
ITGA2B P08514 1/20 0.52
ITGB5 P18084 1/20 0.52
KLK5 Q9Y337 1/20 0.49
CTSS P25774 6/20 0.47
CTSK P43235 5/20 0.47
HDAC8 Q9BY41 1/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPT P10636 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
PTPN1 P18031 3/20 0.45
EPHX2 P34913 1/20 0.44
CTSL P07711 1/20 0.44
CTSB P07858 1/20 0.44
PABPC1 P11940 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561292 0.88 ITGB1 (0.56) ITGB1ITGA4ITGB3ITGAVITGA2B
SCHEMBL14799578 0.88 ITGB1 (0.56) ITGB1ITGA4ITGB3ITGAVITGA2B
SCHEMBL6638467 0.84 ITGB1 (0.63) ITGB1ITGA4ITGB3ITGAVITGA2B
SCHEMBL20715930 0.84 ITGB3 (0.61) ITGB1ITGB3ITGAVITGA2BITGB5
SCHEMBL27278646 0.82 KLK5 (0.54) ITGB1ITGB3ITGAVITGA2BITGB5
SCHEMBL15140552 0.82 ITGB1 (0.48) ITGB1ITGA4ITGB3ITGAVITGA2B
SCHEMBL15140555 0.82 ITGB1 (0.48) ITGB1ITGA4ITGB3ITGAVITGA2B
SCHEMBL19234613 0.81 KLK5 (0.59) ITGB1ITGB3ITGAVITGA2BITGB5
SCHEMBL22427549 0.81 KLK5 (0.53) ITGB1ITGB3ITGAVITGA2BITGB5
SCHEMBL27278632 0.81 KLK5 (0.53) ITGB1ITGB3ITGAVITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6911451-B1 Phenylalanine derivatives CELLTECH R&D LIMITED (GB) 2005-06-28 US disclosed