SCHEMBL6513206

SCHEMBL6513206

CCc1cccc(CC)c1-c1cc(OC(C)C)c(CCC(C)=O)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 12/20 0.41
C5AR1 P21730 1/20 0.40
IAPP P10997 1/20 0.38
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 3/20 0.36
FFAR4 Q5NUL3 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
MEN1 O00255 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
MAPT P10636 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6522026 0.84 S1PR1 (0.41) S1PR1C5AR1CYP2D6CYP2C9SLC6A2
SCHEMBL6514263 0.84 C5AR1 (0.44) S1PR1C5AR1CYP2D6CYP2C9
SCHEMBL1327715 0.79 S1PR1 (0.39) S1PR1C5AR1
SCHEMBL2068766 0.78 C5AR1 (0.39) S1PR1C5AR1CYP2D6CYP2C9LMNA
SCHEMBL2140675 0.76 C5AR1 (0.36) S1PR1C5AR1CYP2D6ALDH1A1SLC6A2
SCHEMBL1328622 0.76 C5AR1 (0.41) S1PR1C5AR1CYP2D6CYP2C9ALDH1A1
SCHEMBL1327704 0.75 C5AR1 (0.38) S1PR1C5AR1CYP2D6CYP2C9MEN1
SCHEMBL1328085 0.74 C5AR1 (0.36) S1PR1C5AR1CYP2D6ALDH1A1MEN1
SCHEMBL1328940 0.74 NPSR1 (0.43) C5AR1FFAR4ALDH1A1MEN1MAPT
SCHEMBL1404966 0.72 ALDH1A1 (0.51) IAPPFFAR4ALDH1A1LMNATAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565452-A2 3-SUBSTITUTED-6-ARYL PYRIDINES AS LIGANDS OF C5A RECEPTORS NEUROGEN CORPORATION (US) 2005-08-24 EP disclosed
WO-2004043925-A2 3-SUBSTITUTED-6-ARYL PYRIDINED AS LIGANDS OF C5A RECEPTORS NEUROGEN CORPORATION (US) 2004-05-27 WO disclosed