SCHEMBL6513231

SCHEMBL6513231

COC(=O)c1ccc(-c2ccc(NCCOCc3ccccc3)cn2)s1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 16/20 0.59
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
CYP3A4 P08684 1/20 0.43
FAAH O00519 1/20 0.43
NR4A2 P43354 1/20 0.40
HPGDS O60760 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5904128 0.89 HDAC1 (0.75) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL5903923 0.87 HDAC1 (0.76) HDAC1CYP3A4FAAHHPGDS
SCHEMBL27615071 0.85 HDAC1 (0.67) HDAC1CYP3A4FAAH
SCHEMBL6197819 0.85 HDAC1 (0.60) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL5903726 0.79 MEN1 (0.59) HDAC1HDAC3HDAC4HDAC8HDAC6
SCHEMBL28942341 0.78 HDAC1 (0.49) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL5903813 0.77 HDAC1 (0.55) HDAC1FAAH
SCHEMBL5904009 0.75 PTPN1 (0.57) HDAC1
SCHEMBL5904123 0.74 HDAC1 (1.00) HDAC1CYP3A4
SCHEMBL5810778 0.74 HDAC1 (0.56) HDAC1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005014588-A1 SUBSTITUTED THIENYL-HYDROXAMIC ACIDS HAVING HISTONE DEACETYLASE ACTIVITY ARGENTA DISCOVERY LIMITED (GB) 2005-02-17 WO disclosed