SCHEMBL6513481

SCHEMBL6513481

CN(CCOc1ccccc1)Cc1ccc(Br)nc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.56
KCNH2 Q12809 1/20 0.50
LTA4H P09960 2/20 0.46
MAOB P27338 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
LMNA P02545 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6507043 0.81 HDAC1 (0.50) TSHRMAOBLMNAKDM4EALDH1A1
SCHEMBL17682060 0.80 TSHR (0.81) TSHRKCNH2LTA4HMAOBMEN1
SCHEMBL11681701 0.78 TSHR (0.68) TSHRKCNH2LTA4HMAOBMEN1
SCHEMBL6513490 0.76 TSHR (0.48) TSHRKCNH2LTA4HMAOBLMNA
SCHEMBL6512171 0.76 SSTR4 (0.41) TSHRLMNAKDM4E
SCHEMBL5255891 0.76 PDCD1 (0.44) LTA4HKDM4EALDH1A1
SCHEMBL22831362 0.75 KCNH2 (0.67) TSHRKCNH2LTA4HALDH1A1CHRNB2
SCHEMBL12854780 0.74 APP (0.52) KCNH2MAOBMEN1KMT2ALMNA
SCHEMBL8430091 0.74 TSHR (0.75) TSHRKCNH2LTA4HMAOBMEN1
SCHEMBL11681713 0.72 TSHR (0.77) TSHRKCNH2LTA4HMAOBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005014588-A1 SUBSTITUTED THIENYL-HYDROXAMIC ACIDS HAVING HISTONE DEACETYLASE ACTIVITY ARGENTA DISCOVERY LIMITED (GB) 2005-02-17 WO disclosed