SCHEMBL6519225

SCHEMBL6519225

O=C(O)c1c(O)[c]ccc1Br

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
TTR P02766 1/20 0.34
DPP4 P27487 1/20 0.33
AKR1C4 P17516 2/20 0.31
AKR1C3 P42330 2/20 0.31
AKR1C2 P52895 2/20 0.31
AKR1C1 Q04828 2/20 0.31
PRNP P04156 1/20 0.30
PTPN2 P17706 1/20 0.30
PTPN1 P18031 1/20 0.30
PTPN6 P29350 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6630310 0.78 CA12 (0.50) CA12CA1CA2CA7CA9
SCHEMBL6633958 0.77 CA1 (0.38) CA12CA1CA2CA7CA9
SCHEMBL30474626 0.71 CA12 (0.43) CA12CA1CA2CA7CA9
SCHEMBL10415958 0.71 CA12 (0.43) CA12CA1CA2CA7CA9
SCHEMBL6519228 0.71 CA12 (0.46) CA12CA1CA2CA7CA9
SCHEMBL6632839 0.71 ALDH1A1 (0.36) CA12CA1CA2CA7CA9
SCHEMBL9732647 0.70
SCHEMBL6255516 0.70
SCHEMBL22097577 0.69 TTR (0.44) CA12CA1CA2CA7CA9
SCHEMBL570378 0.67 CA12 (0.52) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1556375-A2 FLAVONE DERIVATIVES AS INHIBITORS OF CYCLIN-DEPENDENT KINASES Nicholas Piramal India Limited (IN) 2005-07-27 EP disclosed
WO-2004004632-A2 FLAVONE DERIVATIVES AS INHIBITORS OF CYCLIN-DEPENDENT KINASES NICHOLAS PIRAMAL INDIA LIMITED (IN) 2004-01-15 WO disclosed