SCHEMBL6528356

SCHEMBL6528356

Cc1c(C)n(Cc2ccccc2C#N)c(Cl)nc1=O

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 7/20 0.44
KMT2A Q03164 1/20 0.44
GRIN1 Q05586 2/20 0.42
GRIN2B Q13224 2/20 0.42
NOX4 Q9NPH5 1/20 0.42
NPBWR1 P48145 1/20 0.42
CLPP Q16740 1/20 0.41
CYP19A1 P11511 1/20 0.41
MAPK1 P28482 1/20 0.41
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3389261 0.82 DPP4 (0.57) DPP4KMT2AGRIN1GRIN2BNOX4
SCHEMBL3391390 0.78 DPP4 (0.58) DPP4KMT2AGRIN1GRIN2BNOX4
SCHEMBL8438720 0.77 KMT2A (0.53) DPP4KMT2AGRIN1GRIN2BNOX4
SCHEMBL3423901 0.74 DPP4 (0.57) DPP4KMT2ANOX4
SCHEMBL3424634 0.73 KMT2A (0.46) DPP4KMT2AGRIN1GRIN2BNOX4
SCHEMBL16152590 0.73 DPP4 (0.61) DPP4KMT2ANOX4NPBWR1MAPK1
SCHEMBL16201107 0.73 TP53 (0.42) DPP4KMT2AGRIN1GRIN2BNOX4
SCHEMBL3391369 0.72 DPP4 (0.58) DPP4KMT2AGRIN1GRIN2BNOX4
SCHEMBL555383 0.72 DPP4 (0.61) DPP4KMT2ATP53
SCHEMBL3424636 0.72 KMT2A (0.47) DPP4KMT2AGRIN1GRIN2BNOX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016911-A1 4-PYRIMIDONE DERIVATIVES AND THEIR USE AS PEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-02-24 WO disclosed