SCHEMBL8438720

SCHEMBL8438720

Cc1c(C)n(Cc2ccccc2C#N)c(=O)n1Cc1ccccc1C#N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.53
DPP4 P27487 5/20 0.53
NOX4 Q9NPH5 1/20 0.51
ALDH1A1 P00352 4/20 0.50
NPSR1 Q6W5P4 1/20 0.50
C5AR1 P21730 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
CYP19A1 P11511 1/20 0.47
GRIN1 Q05586 1/20 0.47
GRIN2B Q13224 1/20 0.47
EGLN3 Q9H6Z9 1/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
OPRM1 P35372 1/20 0.46
OPRK1 P41145 1/20 0.46
TP53 P04637 1/20 0.45
GALR3 O60755 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8440114 0.87 DPP4 (0.46) KMT2ADPP4NOX4ALDH1A1NPSR1
SCHEMBL8688625 0.86 ALDH1A1 (0.60) KMT2ADPP4NOX4ALDH1A1NPSR1
SCHEMBL8442962 0.85 DPP4 (0.53) KMT2ADPP4NOX4ALDH1A1NPSR1
SCHEMBL8441525 0.84 DPP4 (0.49) KMT2ADPP4NOX4ALDH1A1NPSR1
SCHEMBL17036598 0.79 DPP4 (0.58) KMT2ADPP4NOX4ALDH1A1RXFP1
SCHEMBL8217921 0.79 DPP4 (0.54) KMT2ADPP4NOX4ALDH1A1NPSR1
SCHEMBL6528356 0.77 DPP4 (0.44) KMT2ADPP4NOX4CYP19A1GRIN1
SCHEMBL8216924 0.77 DPP4 (0.64) KMT2ADPP4NOX4ALDH1A1NPSR1
SCHEMBL8443631 0.77 ALDH1A1 (0.55) KMT2ADPP4NOX4ALDH1A1NPSR1
SCHEMBL28406812 0.76 DPP4 (0.58) KMT2ADPP4NOX4RXFP1GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5863914-A ADMINISTERING TO HUMAN N,N-DIMETHYLBENZENE OR N,N-DIMETHYLNAPHTHALENE-CYCLIC UREA DERIVATIVE TO TREAT A DISEASE-STATE CAUSED BY INHIBITION OF FACTOR XA MOHAN RAJU (US) 1999-01-26 US disclosed