Isoquinoline

Isoquinoline

SCHEMBL6529066

c1ccc2cnccc2c1.c1ccc2ncccc2c1.c1ccc2nnccc2c1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
EGFR P00533 1/20 0.42
CYP2A6 P11509 1/20 0.41
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
NPC1 O15118 3/20 0.37
RAB9A P51151 2/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 2/20 0.36
TGFBR1 P36897 1/20 0.35
CASP1 P29466 2/20 0.35
HTT P42858 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
CASP7 P55210 1/20 0.35
KMT2A Q03164 1/20 0.35
NR4A2 P43354 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isoquinoline SCHEMBL1533865 0.93 EGFR (0.56) ALDH1A1EGFRCYP2A6PDGFRBPDGFRA
Isoquinoline SCHEMBL7076555 0.92 EGFR (0.39) ALDH1A1EGFRCYP2A6PDGFRBPDGFRA
Isoquinoline SCHEMBL5027436 0.90 EGFR (0.53) ALDH1A1EGFRCYP2A6PDGFRBPDGFRA
Isoquinoline SCHEMBL1505711 0.90 ALDH1A1 (0.68) ALDH1A1EGFRCYP2A6PDGFRBPDGFRA
Isoquinoline SCHEMBL27938240 0.90 ALDH1A1 (0.68) ALDH1A1EGFRCYP2A6PDGFRBPDGFRA
Quinoline SCHEMBL8074027 0.88 ALDH1A1 (0.71) ALDH1A1EGFRNPC1RAB9APOLB
Quinoline SCHEMBL28191335 0.88 ALDH1A1 (0.71) ALDH1A1EGFRNPC1RAB9APOLB
Isoquinoline SCHEMBL902539 0.86 ALDH1A1 (0.63) ALDH1A1EGFRCYP2A6PDGFRBPDGFRA
Isoquinoline SCHEMBL27889185 0.82 EGFR (0.67) ALDH1A1EGFRCYP2A6PDGFRBPDGFRA
Dipyridyl SCHEMBL27975319 0.82 ALDH1A1 (0.57) ALDH1A1EGFRCYP2A6PDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005121125-A1 ETHER-LINKED HETEROARYL COMPOUNDS PFIZER INC. (US) 2005-12-22 WO disclosed