SCHEMBL6529110

SCHEMBL6529110

CC(C)C[C@H](Nc1nc(NCCc2ccc(S(N)(=O)=O)cc2)nc(Nc2cccc(F)c2)n1)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 19/20 0.60
CA2 P00918 19/20 0.60
CA9 Q16790 19/20 0.60
CA12 O43570 13/20 0.60
CA14 Q9ULX7 13/20 0.60
CA4 P22748 4/20 0.49
CA6 P23280 4/20 0.49
CA7 P43166 4/20 0.49
CA3 P07451 3/20 0.49
CA5A P35218 3/20 0.49
CA13 Q8N1Q1 3/20 0.47
CA5B Q9Y2D0 1/20 0.45
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6529116 1.00 CA1 (0.60) CA1CA2CA9CA12CA14
SCHEMBL6529735 0.92 CA1 (0.52) CA1CA2CA9CA12CA14
SCHEMBL6529732 0.92 CA1 (0.52) CA1CA2CA9CA12CA14
SCHEMBL6530247 0.87 ALDH1A1 (0.47) CA1CA2CA9CA12CA14
SCHEMBL6530426 0.80 ALDH1A1 (0.47) ALDH1A1
SCHEMBL6530423 0.80 ALDH1A1 (0.47) ALDH1A1
SCHEMBL12084421 0.79 CA1 (0.59) CA1CA2CA9CA12CA14
SCHEMBL6529058 0.79 CA1 (0.45) CA1CA2CA9CA12CA4
SCHEMBL12084745 0.78 CA1 (0.58) CA1CA2CA9CA12CA14
SCHEMBL6517091 0.75 QPCT (0.45) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO claimed