SCHEMBL6529152

SCHEMBL6529152

Cc1c(N2CCC(C(N)C(C)(C)C#N)C2)cc(N)c2c(=O)c(C(=O)O)cn(C3CC3)c12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.51
HRH3 Q9Y5N1 1/20 0.41
POLB P06746 2/20 0.39
CACNA1F O60840 1/20 0.39
MAPK1 P28482 1/20 0.39
CACNA1D Q01668 1/20 0.39
CACNA1S Q13698 1/20 0.39
CACNA1C Q13936 1/20 0.39
TOP2A P11388 3/20 0.39
TOP2B Q02880 3/20 0.39
GSK3B P49841 2/20 0.39
ALDH1A1 P00352 2/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6530323 0.91 KCNH2 (0.46) KCNH2HRH3POLBCACNA1FMAPK1
SCHEMBL6527070 0.90 KCNH2 (0.57) KCNH2HRH3POLBCACNA1FMAPK1
SCHEMBL6530311 0.85 KCNH2 (0.61) KCNH2HRH3POLBTOP2ATOP2B
SCHEMBL6529950 0.84 KCNH2 (0.50) KCNH2HRH3POLBCACNA1FMAPK1
SCHEMBL6527770 0.81 KCNH2 (0.77) KCNH2POLBTOP2ATOP2BALDH1A1
SCHEMBL6499864 0.81 KCNH2 (0.53) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL6527941 0.78 KCNH2 (0.79) KCNH2POLBGSK3BALDH1A1CHRM2
SCHEMBL6532564 0.77 KCNH2 (0.60) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL5457708 0.77 KCNH2 (0.35) KCNH2CACNA1C
SCHEMBL5455611 0.76 KCNH2 (0.34) KCNH2CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005049602-A1 QUINOLONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2005-06-02 WO claimed
WO-2005049602-A1 QUINOLONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2005-06-02 WO disclosed