SCHEMBL6529923

SCHEMBL6529923

Cc1ccc2nc(N3CCNCC3)c(-c3ccccc3)c(C)c2c1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.46
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 3/20 0.45
CLK4 Q9HAZ1 2/20 0.45
CYP2D6 P10635 1/20 0.45
TSHR P16473 1/20 0.45
ADRB1 P08588 3/20 0.44
NCF1 P14598 2/20 0.44
HTR6 P50406 1/20 0.43
PRKCI P41743 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CYP2C19 P33261 1/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
HIF1A Q16665 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6529924 0.72 CYP1A2 (0.61) CYP1A2CYP3A4CLK4CYP2D6TSHR
SCHEMBL6770354 0.69 ADRB1 (0.56) CYP1A2CYP3A4CLK4CYP2D6TSHR
SCHEMBL12469779 0.69 HTR2C (0.44) NPY5RCYP1A2CYP3A4CLK4CYP2D6
SCHEMBL2754180 0.69 HRH4 (0.59) NPY5RHRH4
SCHEMBL28610794 0.69 HSD17B10 (0.67) CYP1A2CYP3A4CLK4CYP2D6TSHR
SCHEMBL31652347 0.68 CYP1A2 (0.72) CYP1A2CYP3A4CLK4CYP2D6TSHR
SCHEMBL4472647 0.68 CYP1A2 (0.72) CYP1A2CYP3A4CLK4CYP2D6TSHR
Hydrochloric Acid SCHEMBL30222843 0.68 ADRB1 (0.55) CYP1A2CYP3A4CLK4CYP2D6TSHR
SCHEMBL28111704 0.68 CYP1A2 (0.52) NPY5RCYP1A2CYP3A4CLK4CYP2D6
SCHEMBL27637345 0.67 ESR1 (0.47) CYP1A2CYP3A4TSHRALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005087742-A1 METABOLIC KINASE MODULATORS AND METHODS OF USE AS PESTICIDES EXELIXIS, INC. (US) 2005-09-22 WO claimed
WO-2005087742-A1 METABOLIC KINASE MODULATORS AND METHODS OF USE AS PESTICIDES EXELIXIS, INC. (US) 2005-09-22 WO disclosed