SCHEMBL6530642

SCHEMBL6530642

O=C(Nc1nc2ccccc2n1CCN1CCOCC1)c1ccc(Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 1.00
NPSR1 Q6W5P4 2/20 1.00
OPRK1 P41145 10/20 0.84
OPRM1 P35372 6/20 0.84
OPRD1 P41143 6/20 0.84
HSD17B10 Q99714 3/20 0.84
TSHR P16473 2/20 0.84
MAPK1 P28482 2/20 0.84
LMNA P02545 2/20 0.84
SMN1; SMN2 Q16637 2/20 0.84
HPGD P15428 4/20 0.83
KMT2A Q03164 2/20 0.83
CASP1 P29466 1/20 0.70
CASP7 P55210 1/20 0.70
L3MBTL1 Q9Y468 1/20 0.70
USP2 O75604 2/20 0.68
TP53 P04637 1/20 0.68
RAB9A P51151 1/20 0.68
ALDH1A1 P00352 3/20 0.66
MTOR P42345 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532182 0.87 KDM4E (0.77) KDM4ENPSR1OPRK1OPRM1OPRD1
SCHEMBL6499836 0.85 KDM4E (0.74) KDM4ENPSR1OPRK1OPRM1OPRD1
SCHEMBL11711021 0.84 KDM4E (0.73) KDM4ENPSR1OPRK1OPRM1OPRD1
SCHEMBL16261073 0.83 MTOR (0.74) KDM4ENPSR1OPRK1OPRM1OPRD1
SCHEMBL6529303 0.82 KDM4E (0.69) KDM4ENPSR1OPRK1OPRM1OPRD1
SCHEMBL6505339 0.82 KDM4E (0.69) KDM4ENPSR1OPRK1OPRM1OPRD1
SCHEMBL13500540 0.81 OPRK1 (0.86) KDM4ENPSR1OPRK1OPRM1OPRD1
SCHEMBL3600001 0.81 MTOR (0.70) KDM4ENPSR1OPRK1OPRM1OPRD1
SCHEMBL3598210 0.80 OPRK1 (0.85) KDM4ENPSR1OPRK1OPRM1OPRD1
SCHEMBL3606266 0.80 CLK2 (0.72) KDM4ENPSR1OPRK1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO claimed
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO disclosed