SCHEMBL6532350

SCHEMBL6532350

Cc1cc(C)c(-c2nnc(C(=O)N3CCCC3Br)o2)c(C)c1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 13/20 0.37
HCRTR2 O43614 13/20 0.37
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
TLR9 Q9NR96 2/20 0.33
TLR8 Q9NR97 2/20 0.33
TLR7 Q9NYK1 2/20 0.33
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532310 0.74 NPSR1 (0.49) ALDH1A1HPGD
SCHEMBL6532882 0.73 BTK (0.31)
SCHEMBL6530486 0.70 DPP4 (0.71)
SCHEMBL6529823 0.68 DPP4 (0.51) ALDH1A1HPGD
SCHEMBL14424571 0.61 SMN1; SMN2 (0.32) ALDH1A1HPGDCYP3A4
SCHEMBL5749008 0.58
SCHEMBL12171809 0.58 MYC (0.58) ALDH1A1HPGDCYP3A4
SCHEMBL12171104 0.57 NPC1 (0.62) ALDH1A1HPGDCYP3A4
SCHEMBL28352246 0.57 HPGD (0.55) ALDH1A1HPGD
SCHEMBL8491000 0.57 PDK2 (0.51) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037828-A1 NOVEL INHIBITORS OF DPP-IV, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES LTD. (KR) 2005-04-28 WO disclosed