SCHEMBL6532310

SCHEMBL6532310

Cc1cc(C)c(-c2nnc(C(=O)[C@@H]3CCCN3C(=O)OC(C)(C)C)o2)c(C)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.49
LMNA P02545 1/20 0.49
ALDH1A1 P00352 4/20 0.46
GAA P10253 2/20 0.46
TSHR P16473 2/20 0.46
HSD17B10 Q99714 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 1/20 0.46
GLA P06280 1/20 0.46
HPGD P15428 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.44
EPHX2 P34913 1/20 0.42
MAPT P10636 1/20 0.42
DPP4 P27487 1/20 0.42
DPP8 Q6V1X1 1/20 0.42
DPP7 Q9UHL4 1/20 0.42
NPC1 O15118 1/20 0.41
USP30 Q70CQ3 3/20 0.41
UCHL1 P09936 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6529896 0.81 DPP4 (0.59) NPSR1LMNAALDH1A1GAATSHR
SCHEMBL6532752 0.81 USP30 (0.50) NPSR1LMNAALDH1A1TSHRHSD17B10
SCHEMBL6530486 0.79 DPP4 (0.71) LMNADPP4DPP8DPP7SMN1; SMN2
SCHEMBL6530405 0.78 DPP4 (0.60) NPSR1LMNAALDH1A1GAATSHR
SCHEMBL6530105 0.78 DPP4 (0.60) NPSR1LMNAALDH1A1GAATSHR
SCHEMBL6533469 0.77 HSD17B10 (0.44) NPSR1LMNAALDH1A1GAATSHR
SCHEMBL6532846 0.76 ALDH1A1 (0.50) NPSR1LMNAALDH1A1GAATSHR
SCHEMBL6532278 0.75 PKM (0.52) NPSR1LMNAALDH1A1GAATSHR
SCHEMBL6530822 0.74 DPP4 (0.51) NPSR1LMNAALDH1A1GAATSHR
SCHEMBL6532350 0.74 HCRTR1 (0.37) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037828-A1 NOVEL INHIBITORS OF DPP-IV, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES LTD. (KR) 2005-04-28 WO disclosed