SCHEMBL6534170

SCHEMBL6534170

COc1ccc(-c2cc(Cl)c3ccc(OC)cc3n2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.58
ALDH1A1 P00352 3/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
AURKA O14965 1/20 0.53
AURKB Q96GD4 1/20 0.53
ACACA Q13085 1/20 0.52
LMNA P02545 1/20 0.52
MAPT P10636 1/20 0.52
HPGD P15428 1/20 0.52
HTT P42858 1/20 0.52
SMYD3 Q9H7B4 1/20 0.52
DHODH Q02127 2/20 0.51
PLA2G2A P14555 2/20 0.50
TACR3 P29371 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
ACP1 P24666 2/20 0.48
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6534252 0.94 KDM4E (0.59) KDM4EALDH1A1SMN1; SMN2AURKAAURKB
SCHEMBL6534420 0.93 KDM4E (0.55) KDM4EALDH1A1SMN1; SMN2AURKAAURKB
SCHEMBL5792917 0.91 KDM4E (0.53) KDM4EALDH1A1SMN1; SMN2AURKAAURKB
SCHEMBL374734 0.91 KDM4E (0.72) KDM4EALDH1A1SMN1; SMN2AURKAAURKB
SCHEMBL6534437 0.90 MAPT (0.51) KDM4EALDH1A1SMN1; SMN2AURKAAURKB
SCHEMBL6534218 0.90 KDM4E (0.51) KDM4EALDH1A1SMN1; SMN2AURKAAURKB
SCHEMBL13728214 0.89 ACP1 (0.52) KDM4EALDH1A1SMN1; SMN2AURKAAURKB
SCHEMBL29636809 0.88 KDM4E (0.65) KDM4EALDH1A1SMN1; SMN2AURKAAURKB
SCHEMBL4496204 0.88 KDM4E (0.65) KDM4EALDH1A1SMN1; SMN2AURKAAURKB
SCHEMBL29636789 0.86 MAPT (0.71) KDM4EALDH1A1SMN1; SMN2AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1088818-B1 Quinolin-4-yl derivatives HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6440995-B1 NMDA-RECEPTOR SUBTYPE SELECTIVE BLOCKERS HOFFMAN-LA ROCHE INC. 2002-08-27 US disclosed
EP-1088818-A1 Quinolin-4-yl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-04-04 EP disclosed