SCHEMBL6537494

SCHEMBL6537494

O=C(Nc1cc(F)cc2c(-n3ccnc3)ccnc12)c1c(Cl)cccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CD38 P28907 10/20 0.46
ATR Q13535 2/20 0.43
CYP3A4 P08684 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
JAK2 O60674 3/20 0.42
TYK2 P29597 3/20 0.42
JAK1 P23458 2/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PTGES O14684 1/20 0.40
STING1 Q86WV6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6537403 0.90 CD38 (0.45) CD38ATRCYP3A4CYP1A2CYP2D6
SCHEMBL6537639 0.89 CD38 (0.46) CD38ATRCYP3A4CYP1A2CYP2D6
SCHEMBL6538101 0.88 CYP3A4 (0.46) CD38ATRCYP3A4CYP1A2CYP2D6
SCHEMBL6537488 0.87 CYP3A4 (0.48) CD38ATRCYP3A4CYP1A2CYP2D6
SCHEMBL6538189 0.82 TYK2 (0.51) CYP3A4JAK2TYK2JAK1MEN1
SCHEMBL6537819 0.80 CYP3A4 (0.45) CD38ATRCYP3A4CYP1A2CYP2D6
SCHEMBL6537684 0.80 CYP3A4 (0.48) CD38ATRCYP3A4CYP1A2CYP2D6
SCHEMBL6537943 0.79 CYP3A4 (0.47) CD38ATRCYP3A4CYP1A2CYP2D6
SCHEMBL6537718 0.78 TYK2 (0.50) JAK2TYK2JAK1PTGES
SCHEMBL6538157 0.77 TYK2 (0.39) JAK2TYK2JAK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0876345-B1 HETEROCYCLIC COMPOUNDS AS H+-ATPASES FUJISAWA PHARMACEUTICAL CO (JP) 2004-08-18 EP disclosed
EP-0876345-A1 HETEROCYCLIC COMPOUNDS AS H+-ATPASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-11-11 EP disclosed
WO-1997014681-A1 HETEROCYCLIC COMPOUNDS AS H+-ATPASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-04-24 WO disclosed