SCHEMBL6538940

SCHEMBL6538940

CC(C)(C)OC(=O)N(C[C@@H](O)c1cccc(Cl)c1)[C@H](CO)Cc1ccc(N)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.54
ADRB3 P13945 12/20 0.41
ADRB1 P08588 8/20 0.41
ADRB2 P07550 9/20 0.40
CYP2D6 P10635 2/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
GLA P06280 1/20 0.38
SLC2A1 P11166 2/20 0.38
CYP3A4 P08684 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6539195 1.00 BACE1 (0.54) BACE1ADRB3ADRB1ADRB2CYP2D6
SCHEMBL6538935 1.00 BACE1 (0.54) BACE1ADRB3ADRB1ADRB2CYP2D6
SCHEMBL7120069 0.89 BACE1 (0.43) BACE1ADRB3ADRB1ADRB2CYP2D6
SCHEMBL7120076 0.89 BACE1 (0.43) BACE1ADRB3ADRB1ADRB2CYP2D6
SCHEMBL6478726 0.83 BACE1 (0.52) BACE1ADRB3ADRB1ADRB2CYP2D6
SCHEMBL6478721 0.83 BACE1 (0.52) BACE1ADRB3ADRB1ADRB2CYP2D6
SCHEMBL6539237 0.82 BACE1 (0.52) BACE1ADRB3ADRB1ADRB2GLA
SCHEMBL6539232 0.82 BACE1 (0.52) BACE1ADRB3ADRB1ADRB2GLA
SCHEMBL6478747 0.81 BACE1 (0.50) BACE1ADRB3ADRB1ADRB2CYP2D6
SCHEMBL6478888 0.81 BACE1 (0.48) BACE1ADRB3ADRB1ADRB2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6826033-B2 BETA 3 ADRENERGIC RECEPTOR AGONISTS; TREATMENT OF POLLAKIURIA, URINARY INCONTINENCE, OBESITY OR DIABETES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-11-30 US disclosed
US-20040037022-A1 Aminoalcohol derivatives ASTELLAS PHARMA INC. (JP) 2004-02-26 US disclosed