SCHEMBL6540168

SCHEMBL6540168

COc1ccc(-n2nc(OCC(F)(F)F)cc2-c2ccc(OCCN)cc2)cn1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.44
PTGS1 P23219 7/20 0.44
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
THPO P40225 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
OXTR P30559 1/20 0.37
DYRK3 O43781 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
DYRK1A Q13627 1/20 0.35
DYRK2 Q92630 1/20 0.35
DYRK1B Q9Y463 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5148976 0.99 PTGS2 (0.43) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5148582 0.91 PTGS2 (0.45) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL5152057 0.89 PTGS2 (0.55) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL5148854 0.89 PTGS2 (0.39) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL9996983 0.88 PTGS2 (0.60) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL5148791 0.87 PTGS2 (0.58) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL5148848 0.87 PTGS2 (0.40) PTGS2PTGS1OXTR
SCHEMBL5414201 0.87 PTGS2 (0.41) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5152341 0.86 PTGS2 (0.41) PTGS2PTGS1
Hydrochloric Acid SCHEMBL5149047 0.85 PTGS2 (0.37) PTGS2PTGS1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116475-A1 Pyrazole derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-06-17 US disclosed