SCHEMBL6541879

SCHEMBL6541879

COc1ccc(N2C(OC(=O)O)=C(c3ccc4c(c3)OCO4)c3ccccc3S2(=O)=O)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 10/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
HTT P42858 1/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 1/20 0.39
HSD17B10 Q99714 1/20 0.39
EDNRB P24530 5/20 0.39
HPGD P15428 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6541388 0.90 EDNRA (0.43) EDNRAKDM4EALDH1A1MAPTEDNRB
SCHEMBL6541874 0.88 EDNRA (0.53) EDNRACYP1A2CYP2C9CYP2C19HTT
SCHEMBL6542090 0.86 EDNRA (0.45) EDNRACYP1A2CYP2C9CYP2C19HTT
SCHEMBL6542606 0.86 EDNRA (0.43) EDNRAHTTKDM4EALDH1A1MAPT
SCHEMBL6542684 0.85 EDNRA (0.42) EDNRAKDM4EALDH1A1MAPTHSD17B10
SCHEMBL6542057 0.84 EDNRA (0.51) EDNRAHTTALDH1A1MAPTEDNRB
SCHEMBL6542600 0.83 EDNRA (0.44) EDNRAHTTKDM4EALDH1A1HSD17B10
SCHEMBL6541832 0.83 EDNRA (0.46) EDNRAHTTKDM4EALDH1A1EDNRB
SCHEMBL6542752 0.83 EDNRA (0.49) EDNRAHTTKDM4EALDH1A1MAPT
SCHEMBL7828674 0.82 EDNRA (0.47) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1009743-B1 CERTAIN BENZOTHIAZINE DIOXIDE ENDOTHELIN ANTAGONISTS AND PROCESSES FOR THEIR PREPARATION WARNER LAMBERT CO (US) 2004-06-30 EP claimed