SCHEMBL6548872

SCHEMBL6548872

OC(CON=C(Cl)C=Cc1ccccc1)CN1CCCC1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.55
HSF1 Q00613 8/20 0.51
KDM4E B2RXH2 1/20 0.50
TSHR P16473 2/20 0.49
CYP2D6 P10635 1/20 0.49
HIF1A Q16665 1/20 0.49
RAB9A P51151 1/20 0.44
HSD17B10 Q99714 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
ATM Q13315 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6549930 0.99 ABCB1 (0.57) ABCB1HSF1KDM4ETSHRCYP2D6
SCHEMBL6549925 0.99 ABCB1 (0.57) ABCB1HSF1KDM4ETSHRCYP2D6
SCHEMBL6549086 0.90 POLB (0.51) ABCB1RAB9ASMN1; SMN2MAPK1
SCHEMBL6549091 0.90 POLB (0.51) ABCB1RAB9ASMN1; SMN2MAPK1
SCHEMBL6549255 0.87 HSF1 (0.46) ABCB1HSF1KDM4ETSHRCYP2D6
SCHEMBL6549259 0.87 HSF1 (0.46) ABCB1HSF1KDM4ETSHRCYP2D6
SCHEMBL6548940 0.85 PRMT5 (0.54) SMN1; SMN2
SCHEMBL6548832 0.82 KDM4E (0.60) HSF1KDM4ETSHRCYP2D6
SCHEMBL6548825 0.82 KDM4E (0.60) HSF1KDM4ETSHRCYP2D6
SCHEMBL9329334 0.79 TSHR (0.58) ABCB1KDM4ETSHRCYP2D6HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115697-B1 UNSATURATED HYDROXIMIC ACID DERIVATIVES AS PARP INHIBITORS GENE KUTATO KFT N (HU) 2004-02-04 EP disclosed
US-6500823-B1 ENERGY DEFICIENCY OF THE CELL CAUSED BY PARP INHIBITION, IN DIABETES COMPLICATIONS, IN OXYGEN DEFICIENT STATUS OF THE HEART AND BRAIN, IN NEURODEGENERATIVE DISEASES, IN THE TREATMENT OF AUTOIMMUNE AND/OR VIRAL DISEASES N-GENE RESEARCH LABORATORIES, INC. 2002-12-31 US disclosed
EP-1115697-A1 UNSATURATED HYDROXIMIC ACID DERIVATIVES AS PARP INHIBITORS N-Gene Kutato KFT. (HU) 2001-07-18 EP disclosed
WO-2000014054-A1 UNSATURATED HYDROXIMIC ACID DERIVATIVES AS PARP INHIBITORS N-Gene Kutató Kft. (HU) 2000-03-16 WO disclosed