SCHEMBL6551591

SCHEMBL6551591

O=C(O)CN1CCN(CCCCCCCCCCOc2ccc(C(=O)O)cc2)CCN(CC(=O)O)CCN(CC(=O)O)CC1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 3/20 0.61
HRH3 Q9Y5N1 11/20 0.56
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 2/20 0.55
TP53 P04637 1/20 0.55
TSHR P16473 1/20 0.55
RAB9A P51151 1/20 0.54
PLA2G4B P0C869 1/20 0.54
KCNH2 Q12809 2/20 0.53
HRH1 P35367 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4746238 0.86 HRH3 (0.65) HRH4HRH3KDM4EALDH1A1HRH1
SCHEMBL4746684 0.86 HRH4 (0.55) HRH4HRH3KDM4EALDH1A1TP53
SCHEMBL27457430 0.83 HRH2 (0.60) HRH4HRH3KDM4EALDH1A1TP53
SCHEMBL2087691 0.81 KDM4E (0.72) HRH4HRH3KDM4EALDH1A1RAB9A
SCHEMBL2088353 0.80 KDM4E (0.75) HRH4HRH3KDM4EALDH1A1RAB9A
Hydrochloric Acid SCHEMBL7772340 0.80 KDM4E (0.71) HRH4HRH3KDM4EALDH1A1RAB9A
SCHEMBL10901847 0.80 HRH3 (0.63) HRH3KDM4EALDH1A1KCNH2HRH1
Hydrochloric Acid SCHEMBL4224584 0.79 KDM4E (0.73) HRH4HRH3KDM4EALDH1A1RAB9A
SCHEMBL7911508 0.79 TP53 (0.82) ALDH1A1TP53TSHRPLA2G4B
SCHEMBL2180731 0.79 TP53 (0.82) ALDH1A1TP53TSHRPLA2G4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755385-B1 CHELANT COMPOUNDS AMERSHAM HEALTH AS (NO) 2004-02-11 EP disclosed
US-5798089-A Chelant moieties linked to an aryl moiety by an interrupted alkylene linker NYCOMED SALUTAR, INC. (US) 1998-08-25 US disclosed
EP-0755385-A1 CHELANT COMPOUNDS NYCOMED IMAGING AS (NO) 1997-01-29 EP disclosed
WO-1995028392-A1 CHELANT COMPOUNDS NYCOMED SALUTAR INC. (US) 1995-10-26 WO disclosed