Butenafine

Butenafine

SCHEMBL65526

CN(Cc1ccc(C(C)(C)C)cc1)Cc1cccc2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 1.00
LMNA P02545 4/20 1.00
SLC6A2 P23975 3/20 1.00
SIGMAR1 Q99720 3/20 1.00
ADRA2A P08913 2/20 1.00
NR1I2 O75469 2/20 1.00
HTR2A P28223 2/20 1.00
SLC6A4 P31645 2/20 1.00
KCNH2 Q12809 2/20 1.00
ACHE P22303 1/20 1.00
CYP1A2 P05177 2/20 0.68
CYP2C19 P33261 2/20 0.68
CYP19A1 P11511 1/20 0.58
SQLE Q14534 1/20 0.49
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
HIF1A Q16665 2/20 0.48
DRD2 P14416 1/20 0.48
ADRA2C P18825 1/20 0.48
CNR1 P21554 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butenafine SCHEMBL29354083 1.00 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL20456391 1.00 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL29459249 0.99 LMNA (0.97) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL262301 0.99 LMNA (0.97) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL676912 0.99 LMNA (0.97) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL1648813 0.97 CYP2D6 (0.94) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL500751 0.92 CYP2D6 (0.85) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL9695182 0.89 CYP2D6 (0.80) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL9312678 0.87 CYP2D6 (0.78) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Hydrochloric Acid SCHEMBL9314916 0.86 LMNA (0.76) CYP2D6LMNASLC6A2SIGMAR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 11224 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-20260102419-A1 USE OF COMPOUNDS IN THE TREATMENT OF FUNGAL INFECTIONS BASILEA PHARMACEUTICA INTERNATIONAL AG, ALLSCHWIL (CH) 2026-04-16 US claimed
EP-4719384-A2 COMPOUNDS WITH ANTIFUNGAL PROPERTIES Trustees of Dartmouth College (US) 2026-04-08 EP claimed
US-20260076924-A1 COMPOSITIONS AND METHODS OF TREATMENT FOR TINEA PEDIS THERAPEUTICS INC (US) 2026-03-19 US claimed
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA ATOPIC MEDICAL INC (US) 2026-01-29 US claimed
EP-4676500-A2 MICROBIAL CONSORTIA Kanvas Biosciences, Inc (US) 2026-01-14 EP claimed
US-20260007753-A1 DERMAL SKIN PROTECTANT AND CARRIER INSPIRED MAT STRATEGIES LLC (US) 2026-01-08 US claimed
WO-2025264604-A1 SKIN CARE COMPOSITION AND METHOD OF USING THE SAME THE PROCTER & GAMBLE COMPANY (US) 2025-12-26 WO claimed
US-20250381110-A1 SKIN CARE COMPOSITION AND METHOD OF USING THE SAME PROCTER & GAMBLE (US) 2025-12-18 US claimed
US-12419959-B2 Dermal skin protectant and carrier Inspired Material Strategies, LLC (US) 2025-09-23 US claimed
EP-1024814-A2 USE OF ANTIFUNGAL AGENTS FOR THE TOPICAL TREATMENT OF FUNGUS-INDUCED MUCOSITIS Ponikau, Jens (US) 2000-08-09 EP claimed
WO-1999053913-A1 TOPICAL FORMULATIONS FOR THE TREATMENT OF NAIL FUNGAL DISEASES BERTEK PHARMACEUTICALS, INC. (US) 1999-10-28 WO claimed
WO-1999049895-A2 METHOD FOR INCREASING THE PERMEABILITY OF HORNY HUMAN TISSUE JOHNSON AND JOHNSON CONSUMER COMPANIES, INC. (US) 1999-10-07 WO claimed
WO-1999049835-A1 AN ACIDIFIED COMPOSITION FOR TOPICAL TREATMENT OF NAIL AND SKIN CONDITIONS JOHNSON AND JOHNSON CONSUMER COMPANIES, INC. (US) 1999-10-07 WO claimed
WO-1999020261-A2 USE OF ANTIGUNAL AGENTS FOR THE TOPIAL TREATMENT OF FUNGUS-INDUCED MUCOSITIS PONIKAU JENS (US) 1999-04-29 WO claimed
WO-1997006676-A1 MICROBICIDAL FORMULATIONS BAYER AKTIENGESELLSCHAFT (DE) 1997-02-27 WO claimed
US-5120735-A Synergistic mixture of miconazole, ketoconazole or fluconazole and N-4-tertbutylbenzyl-N-methyl-1-naphthalenemethylamine KAKEN PHARMACEUTICAL CO., LTD. (JP) 1992-06-09 US claimed
EP-0440298-A1 Topical preparations for treating human nails BROCADES PHARMA B.V. (NL) 1991-08-07 EP claimed
EP-0310122-B1 ANTIFUNGAL COMPOSITION KAKEN PHARMACEUTICAL CO., LTD. (JP) 1991-07-24 EP claimed
EP-0310122-A1 Antifungal composition KAKEN PHARMACEUTICAL CO., LTD. (JP) 1989-04-05 EP claimed