SCHEMBL6554049

SCHEMBL6554049

O=C(O)/C=C/c1ccc(-c2nc3c(=O)n(CC4CCCC4)c(=O)n(CC4CCCC4)c3[nH]2)cc1

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 9/20 0.72
ADORA3 P0DMS8 7/20 0.72
ADORA2A P29274 5/20 0.72
ADORA1 P30542 5/20 0.72
RARB P10826 1/20 0.43
PTPN1 P18031 1/20 0.40
MTOR P42345 5/20 0.36
PIK3CA P42336 1/20 0.36
S1PR1 P21453 1/20 0.34
SELP P16109 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6554054 1.00 ADORA2B (0.72) ADORA2BADORA3ADORA2AADORA1RARB
SCHEMBL6555070 0.99 ADORA2B (0.74) ADORA2BADORA3ADORA2AADORA1RARB
SCHEMBL5616732 0.99 ADORA2B (0.74) ADORA2BADORA3ADORA2AADORA1RARB
SCHEMBL6555076 0.99 ADORA2B (0.74) ADORA2BADORA3ADORA2AADORA1RARB
SCHEMBL5616731 0.99 ADORA2B (0.74) ADORA2BADORA3ADORA2AADORA1RARB
Hydrochloric Acid SCHEMBL6554025 0.98 ADORA2B (0.73) ADORA2BADORA3ADORA2AADORA1RARB
SCHEMBL6553545 0.98 ADORA2B (0.69) ADORA2BADORA3ADORA2AADORA1RARB
SCHEMBL6553553 0.98 ADORA2B (0.69) ADORA2BADORA3ADORA2AADORA1RARB
Ethylene SCHEMBL6745653 0.97 ADORA2B (0.74) ADORA2BADORA3ADORA2AADORA1RARB
Ethylene SCHEMBL6745654 0.97 ADORA2B (0.74) ADORA2BADORA3ADORA2AADORA1RARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1104422-B1 PHENYL XANTHINE DERIVATIVES GLAXO GROUP LTD (GB) 2004-02-18 EP disclosed
EP-0775141-B1 PHENYL XANTHINE DERIVATIVES WELLCOME FOUND (GB) 2001-09-26 EP disclosed
EP-0775141-A1 PHENYL XANTHINE DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1997-05-28 EP disclosed
WO-1996004280-A1 PHENYL XANTHINE DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1996-02-15 WO disclosed