SCHEMBL6554152

SCHEMBL6554152

O=c1[nH]c2cc(CC3CC(c4ccc(Cl)cc4)=CCN3)ccc2c2c1CCCC2

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.38
KCNH2 Q12809 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
TNK1 Q13470 2/20 0.36
TNK2 Q07912 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6554106 0.89 PARP1 (0.40) PARP1KCNH2PARP2TNK1TNK2
SCHEMBL6406366 0.73 PARP1 (0.62) PARP1KCNH2PARP2TNK1TNK2
Hydrochloric Acid SCHEMBL6403678 0.71 PARP1 (0.55) PARP1KCNH2PARP2
SCHEMBL6406134 0.71 PARP1 (0.42) PARP1KCNH2PARP2TNK1TNK2
SCHEMBL25093566 0.70 PARP1 (0.51) PARP1KCNH2PARP2
SCHEMBL6554641 0.68 PARP1 (0.53) PARP1KCNH2PARP2
SCHEMBL6556204 0.68 PARP1 (0.53) PARP1KCNH2PARP2TNK1TNK2
SCHEMBL6556334 0.68 PARP1 (0.45) PARP1
SCHEMBL10372460 0.67 CNR1 (0.37)
SCHEMBL6405680 0.67 PARP1 (0.64) PARP1KCNH2PARP2TNK1TNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487800-A1 PHENANTHRIDINONES AS PARP INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-12-22 EP disclosed
WO-2003080581-A1 PHENANTHRIDINONES AS PARP INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-10-02 WO disclosed