SCHEMBL6554240

SCHEMBL6554240

O=c1[nH]c2cc(CN3CCC(c4ccccn4)CC3)ccc2c2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.61
PARP2 Q9UGN5 3/20 0.55
KCNH2 Q12809 2/20 0.55
DRD4 P21917 4/20 0.51
TNK2 Q07912 2/20 0.42
TNK1 Q13470 2/20 0.42
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6405484 0.99 PARP1 (0.60) PARP1PARP2KCNH2DRD4TNK2
SCHEMBL6409266 0.87 PARP1 (0.59) PARP1PARP2KCNH2DRD4TNK2
Hydrochloric Acid SCHEMBL6408219 0.86 PARP1 (0.56) PARP1PARP2KCNH2DRD4TNK2
Hydrochloric Acid SCHEMBL6408278 0.83 PARP1 (0.66) PARP1PARP2KCNH2DRD4DRD2
SCHEMBL6555953 0.80 PARP1 (0.62) PARP1PARP2KCNH2DRD4TNK2
Hydrochloric Acid SCHEMBL6407175 0.79 PARP1 (0.61) PARP1PARP2KCNH2DRD4DRD2
Hydrochloric Acid SCHEMBL6408406 0.79 PARP1 (0.61) PARP1PARP2KCNH2DRD4TNK2
SCHEMBL6554484 0.78 PARP1 (0.66) PARP1PARP2KCNH2
SCHEMBL6406734 0.78 PARP1 (0.77) PARP1PARP2KCNH2
Hydrochloric Acid SCHEMBL6404360 0.78 PARP1 (0.65) PARP1PARP2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487800-A1 PHENANTHRIDINONES AS PARP INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-12-22 EP disclosed
WO-2003080581-A1 PHENANTHRIDINONES AS PARP INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-10-02 WO disclosed