SCHEMBL655582

SCHEMBL655582

COC(=O)c1ccc(C=O)nc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.61
KDM4E B2RXH2 3/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
ALDH1A1 P00352 3/20 0.55
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA12 O43570 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAPT P10636 3/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
KMT2A Q03164 1/20 0.44
ALOX15 P16050 1/20 0.43
ERN1 O75460 1/20 0.43
TSHR P16473 1/20 0.42
XDH P47989 1/20 0.42
HPGDS O60760 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30372051 1.00 MAPK1 (0.61) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL846330 0.84 MAPK1 (0.59) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL846331 0.84 MAPK1 (0.59) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL846377 0.84 MAPK1 (0.59) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL31601570 0.84 MAPK1 (0.59) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL9000473 0.81 MAPK1 (0.56) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL7926743 0.81 CA12 (0.50) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL7389658 0.81 KDM4E (0.57) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL9836119 0.81 CA12 (0.41) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL20419488 0.81 KDM4E (0.64) MAPK1KDM4EL3MBTL1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 351 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113461608-B Synthetic method of 6-formyl methyl nicotinate 江苏弘和药物研发有限公司 2023-03-17 CN claimed
CN-113461608-A Synthetic method of 6-formyl methyl nicotinate 江苏弘和药物研发有限公司 2021-10-01 CN claimed
WO-2008133344-A2 PIPERIDINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-06 WO claimed
US-20080275085-A1 Piperidine derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-06 US claimed
EP-3710428-B1 MODULATORS OF THE INTEGRATED STRESS PATHWAY CALICO LIFE SCIENCES LLC (US) 2026-03-25 EP disclosed
EP-4656201-A2 RAS INHIBITORS Revolution Medicines, Inc. (US) 2025-12-03 EP disclosed
US-20250195521-A1 USE OF SOS1 INHIBITORS TO TREAT MALIGNANCIES WITH SHP2 MUTATIONS Revolution Medicines, Inc. 2025-06-19 US disclosed
CN-115873020-B RAS inhibitors 锐新医药公司 2025-06-13 CN disclosed
US-20250188040-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING WRN HELICASE INHIBITORS VIVIDION THERAPEUTICS INC 2025-06-12 US disclosed
CN-119977956-A 3, 5-Disubstituted-1, 2, 4-triazole compound and preparation method and application thereof 华东师范大学 2025-05-13 CN disclosed
WO-2025095751-A1 NOVEL COMPOUND, AND PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF CANCER COMPRISING SAME 현대약품 주식회사 2025-05-08 WO disclosed
CN-119677716-A Pharmaceutical compositions comprising WRN helicase inhibitors 维维迪恩医疗公司 2025-03-21 CN disclosed
US-5223522-A Anticholesterol agents PFIZER INC. (US) 1993-06-29 US disclosed
EP-0532754-A1 TETRAHYDROIMIDAZOPYRIDINE DERIVATIVE OR ITS SALT YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1993-03-24 EP disclosed
CN-1062263-A The weed killer herbicide that contains the pyridinsulfonamide compounds of replacement ISHIHARA SANGYO KAISHA (JP) 1992-07-01 CN disclosed
US-5120754-A Anticholesterol and antidiabetic agents PFIZER INC. (US) 1992-06-09 US disclosed
CN-1016661-B Herbicidal composition containing pyridine sulfonamide ISHIHARA SANGYO KAISHA (JP) 1992-05-20 CN disclosed
US-5061717-A ANTICHOLESTEROL AGENTS PFIZER INC. (US) 1991-10-29 US disclosed
WO-1989008650-A1 THIAZOLIDINEDIONE HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1989-09-21 WO disclosed
EP-0332331-A2 Thiazolidinedione hypoglycemic agents PFIZER INC. (US) 1989-09-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250195521-A1 USE OF SOS1 INHIBITORS TO TREAT MALIGNANCIES WITH SHP2 MUTATIONS SOS1, PPM1D, PTPN1 MAPK1 202/4885KDM4E 2352/4885L3MBTL1 819/4885
US-20080275085-A1 Piperidine derivative and use thereof TACR2, TACR1, PRLHR MAPK1 1379/4885KDM4E 583/4885L3MBTL1 1776/4885
US-20250188040-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING WRN HELICASE INHIBITORS RECQL, BLM, WRN MAPK1 4017/4885KDM4E 3220/4885L3MBTL1 1538/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.