SCHEMBL6557302

SCHEMBL6557302

CCOc1cc(Cc2cnc(N)nc2N)cc(OCC)c1-c1ccc(CN2CCOCC2)s1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.52
PIK3CA P42336 1/20 0.45
MTOR P42345 1/20 0.45
IKBKE Q14164 1/20 0.43
TBK1 Q9UHD2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557288 0.94 DHFR (0.48) DHFRPIK3CAMTORIKBKETBK1
SCHEMBL6555277 0.94 DHFR (0.46) DHFRPIK3CAMTORIKBKETBK1
SCHEMBL6555373 0.94 DHFR (0.48) DHFR
SCHEMBL6555457 0.91 DHFR (0.43) DHFRPIK3CAMTORIKBKETBK1
SCHEMBL6557155 0.84 DHFR (0.54) DHFR
SCHEMBL6557196 0.83 DHFR (0.55) DHFR
SCHEMBL6555201 0.83 DHFR (0.45) DHFR
SCHEMBL6555139 0.83 DHFR (0.54) DHFR
SCHEMBL6555101 0.82 DHFR (0.52) DHFR
SCHEMBL6555136 0.81 DHFR (0.50) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230224-B1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2004-12-29 EP disclosed
US-6821980-B1 Substituted 5-benzyl-2,4-diaminopyrimidines BASILEA PHARMACEUTICA AG (CH) 2004-11-23 US disclosed