SCHEMBL6557707

SCHEMBL6557707

CCOC(=O)/C(=C/c1ccc(OCCBr)cc1)OCC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.49
PPARG P37231 2/20 0.48
MEN1 O00255 7/20 0.48
KMT2A Q03164 7/20 0.48
MAPT P10636 7/20 0.48
NPSR1 Q6W5P4 3/20 0.48
LMNA P02545 2/20 0.48
MAPK1 P28482 2/20 0.48
S1PR4 O95977 1/20 0.48
S1PR1 P21453 1/20 0.48
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 5/20 0.41
HSP90AA1 P07900 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
MITF O75030 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557711 1.00 NR1H4 (0.49) NR1H4PPARGMEN1KMT2AMAPT
SCHEMBL6409131 0.89 PPARG (0.48) NR1H4PPARGMEN1KMT2AMAPT
SCHEMBL6409133 0.89 PPARG (0.48) NR1H4PPARGMEN1KMT2AMAPT
SCHEMBL14110605 0.89 NR1H4 (0.51) NR1H4MEN1KMT2AMAPTNPSR1
SCHEMBL6055975 0.81 MAPT (0.50) NR1H4MEN1KMT2AMAPTNPSR1
SCHEMBL6055977 0.81 MAPT (0.50) NR1H4MEN1KMT2AMAPTNPSR1
SCHEMBL13916941 0.81 MAPT (0.50) NR1H4MEN1KMT2AMAPTNPSR1
SCHEMBL4217428 0.79 KMT2A (0.73) NR1H4MEN1KMT2AMAPTNPSR1
SCHEMBL4217424 0.79 KMT2A (0.73) NR1H4MEN1KMT2AMAPTNPSR1
SCHEMBL2549286 0.79 MEN1 (0.54) NR1H4MEN1KMT2AMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073643-B1 NEW HETEROCYCLIC COMPOUNDS AND THEIR USE IN MEDICINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM REDDYS LAB LTD DR (IN) 2004-12-29 EP disclosed
EP-1073643-A2 NEW HETEROCYCLIC COMPOUNDS AND THEIR USE IN MEDICINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2001-02-07 EP disclosed
WO-1999008501-A2 NEW HETEROCYCLIC COMPOUNDS AND THEIR USE IN MEDICINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1999-02-25 WO disclosed