Edoxudine

Edoxudine

SCHEMBL65579

CCc1cn([C@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]c1=O

nearest known ligand 0.84

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TK1 P04183 3/20 0.84
TK2 O00142 1/20 0.84
LMNA P02545 2/20 0.72
SMN1; SMN2 Q16637 2/20 0.72
ALOX12 P18054 1/20 0.67
ADRA1A P35348 1/20 0.67
CYP1A2 P05177 1/20 0.65
CYP3A4 P08684 1/20 0.65
TSHR P16473 1/20 0.65
BLM P54132 1/20 0.65
PMP22 Q01453 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Edoxudine SCHEMBL65580 1.00 TK1 (0.84) TK1TK2LMNASMN1; SMN2ALOX12
Edoxudine SCHEMBL9408693 1.00 TK1 (0.84) TK1TK2LMNASMN1; SMN2ALOX12
Edoxudine SCHEMBL1254185 1.00 TK1 (0.84) TK1TK2LMNASMN1; SMN2ALOX12
Edoxudine SCHEMBL21389875 1.00 TK1 (0.84) TK1TK2LMNASMN1; SMN2ALOX12
Edoxudine SCHEMBL12370767 1.00 TK1 (0.84) TK1TK2LMNASMN1; SMN2ALOX12
Edoxudine SCHEMBL5983087 1.00 TK1 (0.84) TK1TK2LMNASMN1; SMN2ALOX12
Edoxudine SCHEMBL5983091 1.00 TK1 (0.84) TK1TK2LMNASMN1; SMN2ALOX12
Edoxudine SCHEMBL11345587 0.95 TK1 (0.78) TK1TK2LMNASMN1; SMN2ALOX12
SCHEMBL13273340 0.92 TK1 (1.00) TK1TK2LMNASMN1; SMN2ALOX12
SCHEMBL5982016 0.92 TK1 (1.00) TK1TK2LMNASMN1; SMN2ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7458 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144879-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS AI-BIOPHARMA (FR) 2026-05-28 US claimed
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
EP-4094767-B1 NUCLEOTIDE AND NUCLEOSIDE THERAPEUTIC COMPOSITIONS AND USES RELATED THERETO UNIV EMORY (US) 2026-05-20 EP claimed
US-20260102422-A1 4'-HALOGEN CONTAINING NUCLEOTIDE AND NUCLEOSIDE THERAPEUTIC COMPOSITIONS AND USES RELATED THERETO UNIV EMORY (US) 2026-04-16 US claimed
US-12595280-B2 Phosphoramidates for the treatment of hepatitis B virus EMORY UNIVERSITY (US) 2026-04-07 US claimed
US-20260092059-A1 Broad Spectrum Antiviral Compositions and Methods EVRYS BIO, LLC (US) 2026-04-02 US claimed
US-20260091068-A1 METHODS FOR TREATING AND PREVENTING DISEASES Tets, Viktor Veniaminovich (US) 2026-04-02 US claimed
EP-3534910-B1 RIFAMPICIN DERIVATIVES WITH ANTIBACTERIAL ACTIVITY POP TEST ONCOLOGY LLC (US) 2026-03-25 EP claimed
US-20260060964-A1 METHODS AND COMPOSITIONS FOR TREATING SEPSIS ANTIVIRUS THERAPEUTICS (US) 2026-03-05 US claimed
WO-2026043843-A1 TETRAHYDROPYRIMIDINE (THP) IONIZABLE LIPIDS FOR EFFICIENT MRNA DELIVERY THE BOARD OF REGENTS OF THE NEVADA SYSTEM OF HIGHER EDUCATION ON BEHALF OF THE UNIVERSITY OF NEVADA, (US) 2026-02-26 WO claimed
WO-1992009287-A1 COMBINATIONS OF VANILLOID COMPOUNDS AND NUCLEOSIDE ANTIVIRAL COMPOUNDS FOR TREATMENT OF HERPES INFECTIONS THE PROCTER & GAMBLE COMPANY (US) 1992-06-11 WO claimed
WO-1992000988-A1 TARGETED DRUG DELIVERY VIA PHOSPHONATE DERIVATIVES BODOR NICHOLAS S (US) 1992-01-23 WO claimed
US-4851391-A TOPICAL GEL ROBUGEN GMBH PHARMAZEUTISCHE FABRIK (DE) 1989-07-25 US claimed
EP-0294443-A1 USE OF NUCLEOSIDES FOR THE MANUFACTURE OF MEDICAMENT FOR TREATMENT OF DISEASES CAUSED BY RETROVIRUS OR HEPATITIS B VIRUS. MEDIVIR AB (SE) 1988-12-14 EP claimed
EP-0277270-A2 N-alkylated quaternary nitrogen-containing heterocycles, process for their preparation and their use in pharmaceutical compositions MEDICEChem.-Pharm. Fabrik Pütter GmbH & Co. KG (DE) 1988-08-10 EP claimed
WO-1988004662-A1 USE OF NUCLEOSIDES FOR THE MANUFACTURE OF MEDICAMENT FOR TREATMENT OF DISEASES CAUSED BY RETROVIRUS OR HEPATITIS B VIRUS Astra Läkemedel Aktiebolag (SE) 1988-06-30 WO claimed
EP-0262344-A2 N-alkylated quaternary nitrogen-containing heterocycles, process for their preparation and their use in pharmaceutical compositions MEDICEChem.-Pharm. Fabrik Pütter GmbH & Co. KG (DE) 1988-04-06 EP claimed
EP-0260428-A2 Cationic surfactants and pharmaceutical compositions containing them MEDICEChem.-Pharm. Fabrik Pütter GmbH & Co. KG (DE) 1988-03-23 EP claimed
EP-0260429-A2 N-alkylated quaternary nitrogen-containing heterocycles, process for their preparation and their use in pharmaceutical compositions MEDICEChem.-Pharm. Fabrik Pütter GmbH & Co. KG (DE) 1988-03-23 EP claimed
EP-0257400-A2 Pharmaceutical compositions containing cationic surfactants MEDICEChem.-Pharm. Fabrik Pütter GmbH & Co. KG (DE) 1988-03-02 EP claimed