SCHEMBL6559013

SCHEMBL6559013

COc1ccc2nc(-c3ccccc3)cc(CCNC(=O)C3CC3)c2c1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 16/20 0.63
MTNR1B P49286 13/20 0.60
ALDH1A1 P00352 1/20 0.57
NQO2 P16083 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6560424 0.87 MTNR1A (0.65) MTNR1AMTNR1B
SCHEMBL6559745 0.85 MTNR1A (0.64) MTNR1AMTNR1BALDH1A1NQO2
SCHEMBL6248773 0.84 MTNR1A (0.75) MTNR1AMTNR1BNQO2
SCHEMBL6559762 0.83 MTNR1A (0.62) MTNR1AMTNR1BNQO2
SCHEMBL6560401 0.80 MTNR1A (0.74) MTNR1AMTNR1BALDH1A1NQO2
SCHEMBL6246356 0.80 MTNR1A (0.80) MTNR1AMTNR1BNQO2
SCHEMBL8961088 0.78 MTNR1A (0.78) MTNR1AMTNR1BALDH1A1NQO2
SCHEMBL8961043 0.78 MTNR1A (0.78) MTNR1AMTNR1BALDH1A1NQO2
SCHEMBL6247137 0.78 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL29493844 0.78 MTNR1A (1.00) MTNR1AMTNR1BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0837850-B1 4-ACYLAMINO(HALOGENO) ALKYL-QUINOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MELATONIN AGONISTS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-09-01 EP disclosed
US-5708005-A MELATONIN RECEPTOR BINDERS, SLEEP DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-13 US disclosed
WO-1997001539-A1 4-ACYLAMINO(HALOGENO) ALKYL-QUINOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MELATONIN AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-16 WO disclosed